Pentaacetylquercetin

Pentaacetylquercetin

SCHEMBL4064499

CC(=O)Oc1cc(OC(C)=O)c2c(=O)c(OC(C)=O)c(-c3ccc(OC(C)=O)c(OC(C)=O)c3)oc2c1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.77
KDM4E B2RXH2 9/20 0.66
CYP3A4 P08684 6/20 0.66
HSD17B10 Q99714 6/20 0.66
MAPT P10636 6/20 0.66
MAPK1 P28482 4/20 0.66
CASP1 P29466 4/20 0.66
CASP7 P55210 4/20 0.66
MEN1 O00255 3/20 0.66
KMT2A Q03164 3/20 0.66
ALOX12 P18054 1/20 0.66
ALDH1A1 P00352 5/20 0.63
CYP2C9 P11712 1/20 0.63
ABCB1 P08183 2/20 0.55
ABCC1 P33527 2/20 0.55
ABCG2 Q9UNQ0 2/20 0.55
TDP1 Q9NUW8 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.53
HPGD P15428 1/20 0.53
GLA P06280 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23278846 0.94 ADORA3 (0.72) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL23483932 0.94 ADORA3 (0.69) ADORA3KDM4ECYP3A4HSD17B10MAPT
Kaempferol Tetraacetate SCHEMBL10379364 0.91 ADORA3 (0.84) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL20581611 0.89 ADORA3 (0.78) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL15965556 0.88 KDM4E (0.66) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL22529297 0.88 ADORA3 (0.61) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL21819719 0.87 ADORA3 (0.72) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL1664667 0.87 ADORA3 (1.00) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL10429428 0.85 ABCG2 (0.77) ADORA3KDM4ECYP3A4HSD17B10MAPT
SCHEMBL5132499 0.85 ADORA3 (0.57) ADORA3KDM4ECYP3A4HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 59 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090130051-A1 Flavonoid Compounds and Uses Thereof HOWARD FLOREY INSTITUTE OF EXPERIMENTAL PHYSIOLOGY AND MEDICINE (AU) 2009-05-21 US claimed
US-12115178-B2 Acylated active agents and methods of their use for the treatment of autoimmune disorders FLAGSHIP PIONEERING INNOVATIONS V, INC. (US) 2024-10-15 US disclosed
EP-3634430-B1 MULTIBIOTIC AGENTS AND METHODS OF USING THE SAME FLAGSHIP PIONEERING INNOVATIONS V INC (US) 2024-08-07 EP disclosed
US-20240180941-A1 ACTIVE AGENTS AND METHODS OF THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS AND NONALCOHOLIC FATTY LIVER DISEASE FLAGSHIP PIONEERING INNOVATIONS V INC (US) 2024-06-06 US disclosed
US-11813272-B2 Active agents and methods of their use for the treatment of metabolic disorders and nonalcoholic fatty liver disease FLAGSHIP PIONEERING INNOVATIONS V, INC. (US) 2023-11-14 US disclosed
US-11813272-B2 Active agents and methods of their use for the treatment of metabolic disorders and nonalcoholic fatty liver disease FLAGSHIP PIONEERING INNOVATIONS V, INC. (US) 2023-11-14 US disclosed
US-11813272-B2 Active agents and methods of their use for the treatment of metabolic disorders and nonalcoholic fatty liver disease FLAGSHIP PIONEERING INNOVATIONS V, INC. (US) 2023-11-14 US disclosed
US-20230293458-A1 MULTIBIOTIC AGENTS AND METHODS OF USING THE SAME FLAGSHIP PIONEERING INNOVATIONS V INC (US) 2023-09-21 US disclosed
US-20230293458-A1 MULTIBIOTIC AGENTS AND METHODS OF USING THE SAME FLAGSHIP PIONEERING INNOVATIONS V INC (US) 2023-09-21 US disclosed
US-20230293458-A1 MULTIBIOTIC AGENTS AND METHODS OF USING THE SAME FLAGSHIP PIONEERING INNOVATIONS V INC (US) 2023-09-21 US disclosed
US-7863323-B1 Flavonols THE UNIVERSITY OF MELBOURNE (AU) 2011-01-04 US disclosed
US-7863323-B1 Flavonols THE UNIVERSITY OF MELBOURNE (AU) 2011-01-04 US disclosed
US-7863323-B1 Flavonols THE UNIVERSITY OF MELBOURNE (AU) 2011-01-04 US disclosed
US-20100226931-A1 Compounds for immunopotentiation NOVARTIS VACCINES AND DIAGNOSTICS, INC. 2010-09-09 US disclosed
US-20100226931-A1 Compounds for immunopotentiation NOVARTIS VACCINES AND DIAGNOSTICS, INC. 2010-09-09 US disclosed
JP-2009096731-A CARBOXYMETHYL ARGININE PRODUCTION INHIBITOR KUMAMOTO UNIV 2009-05-07 JP disclosed
WO-2002020834-A2 METHOD FOR THE IDENTIFICATION OF GENES THAT ARE INVOLVED IN THE MODULATION OF A POPTOSIS IN CELLS EIRX THERAPEUTICS LIMITED (IE) 2002-03-14 WO disclosed
US-6258840-B1 ANTITUMOR AGENTS, ANTIINFLAMMATORY AGENTS, ENZYME INHIBITORS OF KINASES COBRA THERAPEUTICS LIMITED (GB) 2001-07-10 US disclosed
EP-0912541-A1 ANALOGUES OR DERIVATIVES OF QUERCETIN (PRODRUGS) Cobra Therapeutics Limited (GB) 1999-05-06 EP disclosed
WO-1997049693-A1 ANALOGUES OR DERIVATIVES OF QUERCETIN (PRODRUGS) COBRA THERAPEUTICS LIMITED (GB) 1997-12-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11813272-B2 Active agents and methods of their use for the treatment of metabolic disorders and nonalcoholic fatty liver disease FABP1, PYGL, LIPC ADORA3 2284/4885KDM4E 4251/4885CYP3A4 1385/4885
US-20100226931-A1 Compounds for immunopotentiation LY96, ICOS, PDCD1 ADORA3 1365/4885KDM4E 558/4885CYP3A4 1055/4885
US-20240180941-A1 ACTIVE AGENTS AND METHODS OF THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS AND NONALCOHOLIC FATTY LIVER DISEASE FABP1, PYGL, LIPC ADORA3 2284/4885KDM4E 4251/4885CYP3A4 1385/4885
US-20090130051-A1 Flavonoid Compounds and Uses Thereof CAT, NQO1, GPX4 ADORA3 2776/4885KDM4E 4144/4885CYP3A4 518/4885
US-20230293458-A1 MULTIBIOTIC AGENTS AND METHODS OF USING THE SAME SI, FABP2, CEL ADORA3 3910/4885KDM4E 2438/4885CYP3A4 2661/4885
US-12115178-B2 Acylated active agents and methods of their use for the treatment of autoimmune disorders ENPP2, MBOAT7, AADAC ADORA3 3697/4885KDM4E 2430/4885CYP3A4 4519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.