SCHEMBL4093027

SCHEMBL4093027

Cc1cc(C(=O)Nc2n[nH]c3cc(C(=O)NC(C)(C)c4ccccc4)oc23)no1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.44
TP53 P04637 3/20 0.44
USP2 O75604 2/20 0.44
KDM4E B2RXH2 1/20 0.44
GFER P55789 1/20 0.44
AURKA O14965 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 2/20 0.41
NPC1 O15118 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
PTGS2 P35354 1/20 0.40
ALDH1A1 P00352 4/20 0.38
GLA P06280 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4086360 0.87 MAPK1 (0.47) RAB9AAURKANPC1SMN1; SMN2
SCHEMBL4078785 0.87 AURKA (0.42) RAB9ATP53KDM4EAURKAHTT
SCHEMBL4088217 0.86 AURKA (0.51) AURKAHTT
SCHEMBL4082057 0.85 KMT2A (0.44) RAB9ATP53USP2GFERAURKA
SCHEMBL4078482 0.85 HPGD (0.46) RAB9ATP53KDM4EAURKAHTT
SCHEMBL4083114 0.85 AURKA (0.41) RAB9ATP53AURKANPC1SMN1; SMN2
SCHEMBL4088406 0.85 ALDH1A1 (0.47) RAB9ATP53KDM4EAURKANPC1
SCHEMBL4083789 0.84 EGLN1 (0.42) AURKACYP2D6
SCHEMBL4092679 0.84 AURKA (0.49) RAB9AKDM4EAURKANPC1SMN1; SMN2
SCHEMBL4083886 0.83 AURKA (0.44) RAB9ATP53AURKANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed