SCHEMBL412534

SCHEMBL412534

COP(=O)(O)OP(C)(=O)O

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.39
FDPS P14324 1/20 0.35
BLM P54132 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
BTN3A1 O00481 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19057264 0.95 CA2 (0.35) CA2FDPSBLMTDP1
SCHEMBL15831216 0.88 CA2 (0.30) CA2
SCHEMBL10062709 0.84 CA2 (0.47) CA2FDPSBLMTDP1BTN3A1
SCHEMBL1758664 0.84 FDPS (0.41) CA2FDPSBLMTDP1BTN3A1
SCHEMBL13346159 0.82 CA2 (0.39) CA2FDPSBLMTDP1BTN3A1
SCHEMBL13254631 0.81 FDPS (0.39) CA2FDPSBLMTDP1BTN3A1
SCHEMBL24469373 0.80 CA2 (0.37) CA2FDPSBLMTDP1BTN3A1
SCHEMBL889928 0.79 FDPS (0.53) CA2FDPSBLMTDP1BTN3A1
SCHEMBL19387807 0.79 FDPS (0.53) CA2FDPSBLMTDP1BTN3A1
Methyl Phosphonate SCHEMBL28129350 0.78 CA2 (0.57) CA2FDPSBLMTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10040814-B2 Uracyl spirooxetane nucleosides JANSSEN SCIENCES IRELAND UC (IE) 2018-08-07 US disclosed
US-20180099990-A1 URACYL SPIROOXETANE NUCLEOSIDES Janssen Sciences Ireland Unlimited Company (IE) 2018-04-12 US disclosed
US-9845336-B2 Uracyl spirooxetane nucleosides JANSSEN SCIENCES IRELAND UC (IE) 2017-12-19 US disclosed
WO-2017176679-A1 DNA SEQUENCING BY SYNTHESIS WITH NUCLEOTIDE ANALOGUES AND RAMAN DETECTION THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2017-10-12 WO disclosed
US-20170275400-A1 METHOD FOR PREPARING TERMINAL-MODIFIED CONJUGATED DIENE POLYMER, TERMINAL-MODIFIED CONJUGATED DIENE POLYMER, RUBBER COMPOSITION AND TIRE BRIDGESTONE CORPORATION (JP) 2017-09-28 US disclosed
US-20170182181-A1 PHOSPHATE BASED LINKERS FOR INTRACELLULAR DELIVERY OF DRUG CONJUGATES MERCK SHARP & DOHME CORP. (US) 2017-06-29 US disclosed
US-20170145045-A1 URACYL SPIROOXETANE NUCLEOSIDES Janssen Sciences Ireland Unlimited Company (IE) 2017-05-25 US disclosed
US-9657313-B2 Isoprene oligomer, polyisoprene, processes for producing these materials, rubber composition, and pneumatic tire SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2017-05-23 US disclosed
US-9422323-B2 Uracyl spirooxetane nucleosides JANSSEN SCIENCES IRELAND UC (IE) 2016-08-23 US disclosed
US-20160222418-A1 ISOPRENE OLIGOMER, POLYISOPRENE, PROCESSES FOR PRODUCING THESE MATERIALS, RUBBER COMPOSITION, AND PNEUMATIC TIRE SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2016-08-04 US disclosed
US-20140171675-A1 ISOPRENE OLIGOMER, POLYISOPRENE, PROCESSES FOR PRODUCING THESE MATERIALS, RUBBER COMPOSITION, AND PNEUMATIC TIRE YAMAGATA UNIVERSITY (JP) 2014-06-19 US disclosed
US-20130217648-A1 Uracyl Spirooxetane Nucleosides MEDIVIR AB (SE) 2013-08-22 US disclosed
US-8481510-B2 Uracyl spirooxetane nucleosides JANSSEN PRODUCTS, LP (US) 2013-07-09 US disclosed
US-8431588-B2 Cyclopropyl polymerase inhibitors JANSSEN PRODUCTS, LP (US) 2013-04-30 US disclosed
US-8399429-B2 Uracyl cyclopropyl nucleotides JANSSEN PRODUCTS, LP (US) 2013-03-19 US disclosed
US-20120065156-A1 Uracyl Spirooxetane Nucleosides TIBOTEC BVBA (BE) 2012-03-15 US disclosed
US-8030096-B2 Water-soluble rhodamine dyes conjugates APPLIED BIOSYSTEMS LLC (US) 2011-10-04 US disclosed
US-20110230436-A1 Uracyl Cyclopropyl Nucleotides CENTOCOR ORTHO BIOTECH PRODUCTS L.P. (US) 2011-09-22 US disclosed
US-20110092460-A1 CYCLOPROPYL POLYMERASE INHIBITORS CENTOCOR ORTHO BIOTECH PRODUCTS L.P. (US) 2011-04-21 US disclosed
US-20110081688-A1 Water-Soluble Rhodamine Dyes Conjugates Life Technologies Corporation (US) 2011-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170182181-A1 PHOSPHATE BASED LINKERS FOR INTRACELLULAR DELIVERY OF DRUG CONJUGATES CD47, PLPBP, CHERP CA2 1112/4885FDPS 1631/4885BLM 4171/4885
US-20110092460-A1 CYCLOPROPYL POLYMERASE INHIBITORS POLR2E, POLR2H, CTR9 CA2 2778/4885FDPS 2491/4885BLM 2052/4885
US-10040814-B2 Uracyl spirooxetane nucleosides SLC28A1, NUDT1, UMPS CA2 4491/4885FDPS 1100/4885BLM 2873/4885
US-20140171675-A1 ISOPRENE OLIGOMER, POLYISOPRENE, PROCESSES FOR PRODUCING THESE MATERIALS, RUBBER COMPOSITION, AND PNEUMATIC TIRE RCE1, GGPS1, TELO2 CA2 4386/4885FDPS 47/4885BLM 520/4885
US-20120065156-A1 Uracyl Spirooxetane Nucleosides PNP, NUDT1, UMPS CA2 4764/4885FDPS 1365/4885BLM 1859/4885
US-20170145045-A1 URACYL SPIROOXETANE NUCLEOSIDES SLC28A1, NUDT1, UMPS CA2 4491/4885FDPS 1100/4885BLM 2873/4885
US-20160222418-A1 ISOPRENE OLIGOMER, POLYISOPRENE, PROCESSES FOR PRODUCING THESE MATERIALS, RUBBER COMPOSITION, AND PNEUMATIC TIRE RCE1, GGPS1, TELO2 CA2 4386/4885FDPS 47/4885BLM 520/4885
US-20180099990-A1 URACYL SPIROOXETANE NUCLEOSIDES SLC28A1, NUDT1, UMPS CA2 4401/4885FDPS 1034/4885BLM 3012/4885
US-20130217648-A1 Uracyl Spirooxetane Nucleosides PNP, NUDT1, UMPS CA2 4764/4885FDPS 1365/4885BLM 1859/4885
US-20110230436-A1 Uracyl Cyclopropyl Nucleotides NUDT1, PNP, RNGTT CA2 4567/4885FDPS 1228/4885BLM 2308/4885
US-20110081688-A1 Water-Soluble Rhodamine Dyes Conjugates SLC43A3, ABCG2, TARBP1 CA2 3116/4885FDPS 3392/4885BLM 1548/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.