Guanosine

Guanosine

SCHEMBL413586

Nc1nc2c(ncn2[C@@H]2O[C@H](CO)C(O)[C@@H]2O)c(=O)[nH]1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.76
HINT1 P49773 4/20 0.68
NT5E P21589 2/20 0.68
PNP P00491 1/20 0.65
PAX8 Q06710 1/20 0.65
GSK3A P49840 2/20 0.64
RPS6KA3 P51812 2/20 0.64
MAPK14 Q16539 2/20 0.64
TGM2 P21980 1/20 0.62
LMNA P02545 1/20 0.62
HIF1A Q16665 1/20 0.62
ADORA2A P29274 3/20 0.62
ADORA3 P0DMS8 1/20 0.62
ADORA2B P29275 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guanosine SCHEMBL34912 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL8593215 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL531207 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL24049416 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL11986902 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL24049608 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL24049417 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL24049467 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL20750695 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8
Guanosine SCHEMBL16800938 1.00 HPGD (0.76) HPGDHINT1NT5EPNPPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 226 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11753431-B2 Compounds comprising cleavable linker and uses thereof INTOCELL, INC. (KR) 2023-09-12 US disclosed
US-11753431-B2 Compounds comprising cleavable linker and uses thereof INTOCELL, INC. (KR) 2023-09-12 US disclosed
US-20230174567-A1 SYNTHESIS OF FLUORINATED NUCLEOTIDES MERCK SHARP & DOHME LLC (US) 2023-06-08 US disclosed
US-20210388017-A1 COMPOUNDS COMPRISING CLEAVABLE LINKER AND USES THEREOF INTOCELL, INC. (KP) 2021-12-16 US disclosed
EP-3505176-A1 MODIFIED POLYNUCLEOTIDES FOR THE PRODUCTION OF SECRETED PROTEINS Moderna Therapeutics, Inc. (US) 2019-07-03 EP disclosed
EP-3501550-A1 MODIFIED POLYNUCLEOTIDES FOR THE PRODUCTION OF PROTEINS ASSOCIATED WITH HUMAN DISEASE Moderna Therapeutics, Inc. (US) 2019-06-26 EP disclosed
WO-2019008441-A1 COMPOUNDS COMPRISING CLEAVABLE LINKER AND USES THEREOF INTOCELL, INC. (KR) 2019-01-10 WO disclosed
US-20180170990-A1 MODIFIED POLYNUCLEOTIDES FOR THE PRODUCTION OF NUCLEAR PROTEINS MODERNATX, INC. 2018-06-21 US disclosed
US-20180125937-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE, AND NUCLEIC ACID COMPOSITIONS MODERNATX, INC. (US) 2018-05-10 US disclosed
US-20180086807-A1 MODIFIED POLYNUCLEOTIDES FOR THE PRODUCTION OF PROTEINS ASSOCIATED WITH HUMAN DISEASE MODERNATX, INC. 2018-03-29 US disclosed
WO-2013090648-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE, AND NUCLEIC ACID COMPOSITIONS modeRNA Therapeutics (US) 2013-06-20 WO disclosed
US-20130156849-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE, AND NUCLEIC ACID COMPOSITIONS modeRNA Therapeutics (US) 2013-06-20 US disclosed
US-20130123481-A1 MODIFIED NUCLEOSIDES, NUCLEOTIDES, AND NUCLEIC ACIDS, AND USES THEREOF modeRNA Therapeutics (US) 2013-05-16 US disclosed
US-20130115272-A1 MODIFIED NUCLEOSIDES, NUCLEOTIDES, AND NUCLEIC ACIDS, AND USES THEREOF modeRNA Therapeutics (US) 2013-05-09 US disclosed
US-20130115272-A1 MODIFIED NUCLEOSIDES, NUCLEOTIDES, AND NUCLEIC ACIDS, AND USES THEREOF modeRNA Therapeutics (US) 2013-05-09 US disclosed
US-20130102655-A1 ALKYNYL-DERIVATIZED CAP ANALOGS, PREPARATION AND USES THEREOF Life Technologies Corporation (US) 2013-04-25 US disclosed
WO-2013052523-A1 MODIFIED NUCLEOSIDES, NUCLEOTIDES, AND NUCLEIC ACIDS, AND USES THEREOF modeRNA Therapeutics (US) 2013-04-11 WO disclosed
US-20130052710-A1 RNA INCLUDING NUCLEOSIDE COMPOUND, METHOD FOR REGULATING AMOUNT OF PROTEIN PRODUCED FROM THE RNA, AND NUCLEOSIDE COMPOUND RIKEN (JP) 2013-02-28 US disclosed
US-20120065386-A1 SYNTHESIS OF LABILE BASE PROTECTED - MODIFIED DEOXY & MODIFIED RIBO NUCLEOSIDES, CORRESPONDING PHOSPHORAMIDITES AND SUPPORTS AND THEIR USE IN HIGH PURITY OLIGONUCLEOTIDE SYNTHESIS CHEMGENES CORPORATION 2012-03-15 US disclosed
US-7919446-B1 Post-CMP cleaning compositions and methods of using same INTERMOLECULAR, INC. (US) 2011-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123481-A1 MODIFIED NUCLEOSIDES, NUCLEOTIDES, AND NUCLEIC ACIDS, AND USES THEREOF ADAR, NT5C3B, NSUN2 HPGD 2978/4885HINT1 121/4885NT5E 10/4885
US-20180170990-A1 MODIFIED POLYNUCLEOTIDES FOR THE PRODUCTION OF NUCLEAR PROTEINS POLN, POLRMT, MSH2 HPGD 3220/4885HINT1 2405/4885NT5E 718/4885
US-20120065386-A1 SYNTHESIS OF LABILE BASE PROTECTED - MODIFIED DEOXY & MODIFIED RIBO NUCLEOSIDES, CORRESPONDING PHOSPHORAMIDITES AND SUPPORTS AND THEIR USE IN HIGH PURITY OLIGONUCLEOTIDE SYNTHESIS RNMT, POLRMT, RNGTT HPGD 1464/4885HINT1 494/4885NT5E 324/4885
US-20180125937-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE, AND NUCLEIC ACID COMPOSITIONS NSUN2, RNMT, NSUN3 HPGD 3755/4885HINT1 440/4885NT5E 44/4885
US-20130156849-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE, AND NUCLEIC ACID COMPOSITIONS NSUN2, RNMT, NSUN3 HPGD 3755/4885HINT1 440/4885NT5E 44/4885
US-20130102655-A1 ALKYNYL-DERIVATIZED CAP ANALOGS, PREPARATION AND USES THEREOF RNGTT, RNMT, NSUN3 HPGD 4494/4885HINT1 335/4885NT5E 1269/4885
US-20210388017-A1 COMPOUNDS COMPRISING CLEAVABLE LINKER AND USES THEREOF VIP, ANTXR2, TNFRSF9 HPGD 2968/4885HINT1 3537/4885NT5E 1350/4885
US-11753431-B2 Compounds comprising cleavable linker and uses thereof VIP, ANTXR2, TNFRSF9 HPGD 2968/4885HINT1 3537/4885NT5E 1350/4885
US-20180086807-A1 MODIFIED POLYNUCLEOTIDES FOR THE PRODUCTION OF PROTEINS ASSOCIATED WITH HUMAN DISEASE POLRMT, POLM, POLN HPGD 3640/4885HINT1 2055/4885NT5E 874/4885
US-20130052710-A1 RNA INCLUDING NUCLEOSIDE COMPOUND, METHOD FOR REGULATING AMOUNT OF PROTEIN PRODUCED FROM THE RNA, AND NUCLEOSIDE COMPOUND RNMT, NSUN2, RNGTT HPGD 3670/4885HINT1 252/4885NT5E 323/4885
US-20230174567-A1 SYNTHESIS OF FLUORINATED NUCLEOTIDES NUDT1, NT5C3B, MTAP HPGD 505/4885HINT1 46/4885NT5E 21/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.