Iomazenil

Iomazenil

SCHEMBL41658

CCOC(=O)c1ncn2c1CN(C)C(=O)c1c(I)cccc1-2

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 13/20 0.71
GABRG2 P18507 12/20 0.71
GABRB3 P28472 12/20 0.71
GABRA5 P31644 12/20 0.71
GABRA3 P34903 12/20 0.71
GABRA2 P47869 12/20 0.71
GABRA6 Q16445 8/20 0.62
GABRB2 P47870 7/20 0.62
GABRA4 P48169 3/20 0.61
ALDH1A1 P00352 2/20 0.61
MEN1 O00255 1/20 0.61
GABRP O00591 1/20 0.61
GABRD O14764 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
TSHR P16473 1/20 0.61
GABRB1 P18505 1/20 0.61
CYP2C19 P33261 1/20 0.61
GABRE P78334 1/20 0.61
KMT2A Q03164 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iomazenil SCHEMBL29385986 1.00 GABRA1 (0.71) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7334382 0.91 GABRA1 (0.75) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10365966 0.89 GABRA1 (0.72) GABRA1GABRG2GABRB3GABRA5GABRA3
Sarmazenil SCHEMBL195304 0.88 GABRA1 (0.71) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7329697 0.88 GABRA1 (0.71) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9745968 0.88 GABRA1 (0.71) GABRA1GABRG2GABRB3GABRA5GABRA3
Iomazenil (123I) SCHEMBL17022271 0.88 GABRA1 (0.71) GABRA1GABRG2GABRB3GABRA5GABRA3
Iomazenil (123I) SCHEMBL29374678 0.88 GABRA1 (0.71) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10627713 0.87 GABRA1 (0.70) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL11887388 0.86 GABRA1 (0.68) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 215 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230405018-A1 FLUMAZENIL FORMULATIONS FOR SUBCUTANEOUS INJECTION AND METHODS OF TREATMENT USING GABA RECEPTOR MODULATORS BEXSON BIOMEDICAL, INC. 2023-12-21 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-0353754-B1 RADIOACTIVELY MARKED BENZODIAZEPIN DERIVATES F. HOFFMANN-LA ROCHE AG (CH) 1992-12-02 EP claimed
US-20260137765-A1 METHODS OF PRODUCING SHIGA TOXIN B-SUBUNIT (STXB) MONOMERS AND OLIGOMERS, AND USES THEREOF INSTITUT CURIE (FR) 2026-05-21 US disclosed
EP-3129065-B1 TARGETED DRUG DELIVERY THROUGH AFFINITY BASED LINKERS AKAMARA THERAPEUTICS INC (US) 2026-05-13 EP disclosed
US-12527854-B2 Methods of producing Shiga toxin B-subunit (STxB) monomers and oligomers, and uses thereof INSTITUT CURIE (FR) 2026-01-20 US disclosed
US-20250367232-A1 HALOGEN TREATMENT OF HEART ATTACK AND ISCHEMIC INJURY HUTCHINSON FRED CANCER RES (US) 2025-12-04 US disclosed
US-20250281535-A1 ANTI-HUMAN CD45RC BINDING DOMAINS AND USES THEREOF ABOLERIS PHARMA (FR) 2025-09-11 US disclosed
EP-4401842-B1 ANTI-HUMAN CD45RC BINDING DOMAINS AND USES THEREOF ABOLERIS PHARMA (FR) 2025-08-27 EP disclosed
WO-2001089586-A2 TC AND RE CARBONYL COMPLEXES FOR PERTECHNETATE AND PERRHENATE MALLINCKRODT INC. (US) 2001-11-29 WO disclosed
WO-2001000637-A1 GROUP (VII) TRANSITION-METAL COMPLEXES WITH MULTIDENTATE AMINOPOLYCARBOXYLATE LIGANDS AND A KIT FOR PRODUCING THEM MALLINCKRODT INC. (US) 2001-01-04 WO disclosed
EP-1019095-A1 METHOD FOR THE PREPARATION OF FACIAL METAL TRICARBONYL COMPOUNDS AND THEIR USE IN THE LABELLING OF BIOLOGICALLY ACTIVE SUBSTRATES Mallinckrodt Inc. (US) 2000-07-19 EP disclosed
EP-0879606-A1 Method for the preparation of facial metal tricarbonyl compounds and their use in the labelling of biologically active substrates PAUL SCHERRER INSTITUT (CH) 1998-11-25 EP disclosed
WO-1998048848-A1 METHOD FOR THE PREPARATION OF FACIAL METAL TRICARBONYL COMPOUNDS AND THEIR USE IN THE LABELLING OF BIOLOGICALLY ACTIVE SUBSTRATES MALLINCKRODT INC. (US) 1998-11-05 WO disclosed
US-5096695-A Diagnosis of brain disorders, cardiovascular diseases, epilepsy, psychosis HOFFMANN-LAROCHE INC. (US) 1992-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12527854-B2 Methods of producing Shiga toxin B-subunit (STxB) monomers and oligomers, and uses thereof STXBP1, RNGTT, UPF1 GABRA1 879/4885GABRG2 1092/4885GABRB3 387/4885
US-20230405018-A1 FLUMAZENIL FORMULATIONS FOR SUBCUTANEOUS INJECTION AND METHODS OF TREATMENT USING GABA RECEPTOR MODULATORS GABBR1, GABBR2, GABRB2 GABRA1 8/4885GABRG2 14/4885GABRB3 9/4885
US-20260137765-A1 METHODS OF PRODUCING SHIGA TOXIN B-SUBUNIT (STXB) MONOMERS AND OLIGOMERS, AND USES THEREOF STXBP1, HBB, UPF1 GABRA1 1184/4885GABRG2 1329/4885GABRB3 342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.