SCHEMBL418126

SCHEMBL418126

Cn1c(C(=O)O)cc2cc(Br)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 1.00
KDM4E B2RXH2 2/20 0.66
ALDH1A1 P00352 2/20 0.66
HPGD P15428 2/20 0.66
HSD17B10 Q99714 2/20 0.66
SMN1; SMN2 Q16637 1/20 0.62
GPR35 Q9HC97 1/20 0.57
GFER P55789 1/20 0.52
SRD5A2 P31213 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16440985 0.86 MCL1 (0.76) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL6752295 0.86 MCL1 (0.76) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3534182 0.85 MCL1 (0.73) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL1096760 0.82 L3MBTL1 (0.70) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL31435640 0.82 MCL1 (0.69) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL10084917 0.82 MCL1 (0.69) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL5599830 0.81 KDM4E (0.68) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2001537 0.81 HSD17B10 (0.68) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL30547707 0.81 KDM4E (0.68) MCL1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL5889548 0.81 KDM4E (0.68) MCL1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4651872-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE TO TREAT HYPOPARATHYROIDISM AND OSTEOPOROSIS Septerna, Inc. (US) 2025-11-26 EP disclosed
WO-2024155601-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE TO TREAT HYPOPARATHYROIDISM AND OSTEOPOROSIS SEPTERNA, INC. (US) 2024-07-25 WO disclosed
WO-2023226950-A1 PEPTIDOMIMETIC STAT PROTEIN DEGRADER, COMPOSITION AND USE THEREOF 杭州和正医药有限公司 2023-11-30 WO disclosed
CN-117126231-A Peptoid STAT protein degradation agent, composition and application thereof 杭州和正医药有限公司 2023-11-28 CN disclosed
CN-114702504-B Trifluoromethyl substituted indolopyranone compound, preparation method thereof and application thereof in antitumor drugs 平顶山学院 2023-04-07 CN disclosed
CN-114702504-A Trifluoromethyl substituted indolopyranone compound, preparation method thereof and application thereof in antitumor drugs 平顶山学院 2022-07-05 CN disclosed
EP-3400210-B1 \"MULTI-TARGET\" COMPOUNDS WITH INHIBITORY ACTIVITY TOWARDS HISTONE DEACETYLASES AND TUBULIN POLYMERISATION, FOR USE IN THE TREATMENT OF CANCER UNIV PARIS SACLAY (FR) 2021-09-29 EP disclosed
EP-2607348-B1 Plasminogen Activator Inhibitor-1 Inhibitor RENASCIENCE INC (JP) 2021-03-17 EP disclosed
CN-109705071-A Hdac inhibitor and its preparation method and application 成都先导药物开发有限公司 2019-05-03 CN disclosed
EP-3400210-A2 \"MULTI-TARGET\" COMPOUNDS WITH INHIBITORY ACTIVITY TOWARDS HISTONE DEACETYLASES AND TUBULIN POLYMERISATION, FOR USE IN THE TREATMENT OF CANCER Universite Paris-Sud (FR) 2018-11-14 EP disclosed
US-7544803-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2009-06-09 US disclosed
US-7544803-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2009-06-09 US disclosed
US-20080249126-A1 1,3-SUBSTITUTED CYCLOALKYL DERIVATIVES HAVING ACIDIC, MOSTLY HETEROCYCLIC GROUPS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-10-09 US disclosed
US-20080249126-A1 1,3-SUBSTITUTED CYCLOALKYL DERIVATIVES HAVING ACIDIC, MOSTLY HETEROCYCLIC GROUPS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-10-09 US disclosed
US-6989384-B2 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis AGOURON PHARMACEUTICALS, INC. (US) 2006-01-24 US disclosed
US-20050165049-A1 Vanilloid receptor ligands and their use in treatments AMGEN, INC. 2005-07-28 US disclosed
US-20050080121-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis AGOURON PHARMACEUTICALS, INC. 2005-04-14 US disclosed
CN-1525957-A Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis ������ҩ�����޹�˾ 2004-09-01 CN disclosed
US-6632825-B2 Picornaviral 3C protease enzyme inhibitors; amide ester or amide acid derivatives AGOURON PHARMACEUTICALS, INC. 2003-10-14 US disclosed
US-20020061916-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis AGOURON PHARMACEUTICALS, INC. 2002-05-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080249126-A1 1,3-SUBSTITUTED CYCLOALKYL DERIVATIVES HAVING ACIDIC, MOSTLY HETEROCYCLIC GROUPS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS GPR119, PC, FFAR1 MCL1 2050/4885KDM4E 4119/4885ALDH1A1 242/4885
US-20050165049-A1 Vanilloid receptor ligands and their use in treatments TRPV1, TRPV2, TRPV3 MCL1 1264/4885KDM4E 4218/4885ALDH1A1 3253/4885
US-20050080121-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis PRCP, RNPEP, SARNP MCL1 3640/4885KDM4E 3080/4885ALDH1A1 4076/4885
US-20020061916-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis PRCP, RNASEL, RNASEH1 MCL1 3478/4885KDM4E 3119/4885ALDH1A1 3499/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.