SCHEMBL4192960

SCHEMBL4192960

COC(=O)C1=C(C(=O)OC)C2C=CC1C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 7/20 0.42
TSHR P16473 2/20 0.38
NPSR1 Q6W5P4 1/20 0.37
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA12 O43570 3/20 0.37
CA7 P43166 3/20 0.37
CA9 Q16790 3/20 0.37
CA14 Q9ULX7 3/20 0.37
TDP1 Q9NUW8 2/20 0.37
GAA P10253 2/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
NFKB1 P19838 1/20 0.35
XDH P47989 1/20 0.35
GFER P55789 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
FUT7 Q11130 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13947949 0.92 SLC6A3 (0.38) SLC6A3TSHRCA1CA2CA12
SCHEMBL11583334 0.87 SLC6A3 (0.41) SLC6A3TSHRTDP1GAALMNA
SCHEMBL11526468 0.87 ADORA3 (0.47) SLC6A3TSHRNPSR1GAAKDM4E
SCHEMBL15586518 0.86 HSD17B10 (0.39) SLC6A3TSHRNPSR1CA1CA2
SCHEMBL12395334 0.86 SLC6A3 (0.37) SLC6A3TSHRNPSR1CA1CA2
SCHEMBL11529327 0.82 SLC6A3 (0.36) SLC6A3TSHRNPSR1TDP1GAA
SCHEMBL11525443 0.81 MAPK1 (0.37)
SCHEMBL11527344 0.80 CNR1 (0.34) SLC6A3TSHRL3MBTL1HSD17B10
SCHEMBL11524398 0.78 SLC6A3 (0.52) SLC6A3TSHRLMNASMN1; SMN2
SCHEMBL11531802 0.78 SLC6A3 (0.39) SLC6A3NPSR1KDM4EHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 98 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130150613-A1 SYNTHESIS OF HALF ESTERS TIMES THREE WIRELESS, INC. (CA) 2013-06-13 US claimed
US-4582578-A Method for the electrochemical conversion of a quadricyclane to a norbornadiene REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1986-04-15 US claimed
EP-3893889-B1 THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF TERNS INC (US) 2026-01-28 EP disclosed
US-20260001867-A1 THR BETA RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF TERNS PHARMACEUTICALS, INC. 2026-01-01 US disclosed
US-12459926-B2 THRβ receptor agonist compound and preparation method and use thereof Terns, Inc. (US) 2025-11-04 US disclosed
US-12365669-B2 THRβ receptor agonist compound and preparation method and use thereof Terns, Inc. (US) 2025-07-22 US disclosed
EP-4574821-A1 THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF Terns, Inc. (US) 2025-06-25 EP disclosed
US-12338232-B2 THRβ receptor agonist compound and preparation method and use thereof Terns, Inc. (US) 2025-06-24 US disclosed
US-20250179053-A1 THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF TERNS PHARMACEUTICALS, INC. 2025-06-05 US disclosed
US-20250179054-A1 THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF TERNS PHARMACEUTICALS, INC. 2025-06-05 US disclosed
EP-4529954-A2 THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF Terns, Inc. (US) 2025-04-02 EP disclosed
US-5081088-A Preparing propylene polymers BASF AKTIENGESELLSCHAFT (DE) 1992-01-14 US disclosed
US-4132750-A RING OPENING POLYMERIZATION OF NORBORNENE DERIVATIVES SHOWA DENKO K.K. (JP) 1979-01-02 US disclosed
US-4105608-A HIGH IMPACT COMPOSITION OF RING-OPENING POLYMERIZATION PRODUCT SHOWA DENKO K.K. (JP) 1978-08-08 US disclosed
US-4080491-A CATALYST CONTAINS ORGANOMETALLIC COMPOUND AND THE REACTION PRODUCT OF TUNGSTEN OR MOLYBDENUM OXIDE AND A PHOSPHOROUS HALIDE OR OXYHALIDE SHOWA DENKO K.K. (JA) 1978-03-21 US disclosed
US-4059561-A AND A HALOGEN COMPOUND SHOWA DENKO KABUSHIKI KAISHA (JA) 1977-11-22 US disclosed
US-4028482-A LOW VISCOSITY POLYALKENAMER SHOWA DENKO KABUSHIKI KAISHA (JA) 1977-06-07 US disclosed
US-4022954-A ADHESIVES, FLOCCULATING AGENTS, ION EXCHANGE RESINS, MOLDING AGENTS SHOWA DENKO KABUSHIKI KAISHA (JA) 1977-05-10 US disclosed
US-3991139-A NORBORNENE DERIVATIVES, PHENOLS, ESTER THIOETHERS SHOWA DENKO KABUSHIKI KAISHA (JA) 1976-11-09 US disclosed
US-3959234-A CATALYSTS OF ORGANOALUMINUM COMPOUNDS AND A TUNGSTEN OR MOLYBDENUM COMPOUND, RING-OPENING SHOWA DENKO KABUSHIKI KAISHA (JA) 1976-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179054-A1 THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF THRB, THRA, TRHR SLC6A3 850/4885TSHR 4/4885NPSR1 99/4885
US-20260001867-A1 THR BETA RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF THRB, THRA, ADRB1 SLC6A3 1083/4885TSHR 15/4885NPSR1 286/4885
US-20250179053-A1 THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF THRB, THRA, TRHR SLC6A3 850/4885TSHR 4/4885NPSR1 99/4885
US-12459926-B2 THRβ receptor agonist compound and preparation method and use thereof THRB, THRA, TRHR SLC6A3 854/4885TSHR 4/4885NPSR1 85/4885
US-12365669-B2 THRβ receptor agonist compound and preparation method and use thereof THRB, THRA, TRHR SLC6A3 854/4885TSHR 4/4885NPSR1 85/4885
US-20130150613-A1 SYNTHESIS OF HALF ESTERS BCKDK, CES1, KHK SLC6A3 4622/4885TSHR 3847/4885NPSR1 2548/4885
US-12338232-B2 THRβ receptor agonist compound and preparation method and use thereof THRB, THRA, TRHR SLC6A3 854/4885TSHR 4/4885NPSR1 85/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.