SCHEMBL420855

SCHEMBL420855

CC(C)(C)[Si](C)(C)OCC1CCC(=O)C1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 1/20 0.37
TOP2A P11388 3/20 0.35
DUT P33316 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9606663 1.00 FKBP1A (0.37) FKBP1ATOP2ADUT
SCHEMBL30106079 1.00 FKBP1A (0.37) FKBP1ATOP2ADUT
SCHEMBL420544 0.90 FKBP1A (0.36) FKBP1ATOP2ADUT
SCHEMBL11970804 0.86 TOP2A (0.38) FKBP1ATOP2ADUT
SCHEMBL19783450 0.84 DUT (0.33) DUT
SCHEMBL7790340 0.78 DUT (0.35) DUT
SCHEMBL15570491 0.77 FKBP1A (0.32) FKBP1A
SCHEMBL8972926 0.76 IRAK4 (0.35) FKBP1ATOP2ADUT
SCHEMBL20660408 0.76 IRAK4 (0.35) FKBP1ATOP2ADUT
SCHEMBL8062803 0.76 FKBP1A (0.33) FKBP1ATOP2ADUT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250263390-A1 NOVEL SUBSTITUTED 6,7-DIHYDRO-5H-BENZO[7]ANNULENE COMPOUNDS AND THEIR DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF SANOFI (FR) 2025-08-21 US disclosed
EP-4508030-A1 SUBSTITUTED 6,7-DIHYDRO-5H-BENZO[7]ANNULENE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF Sanofi (FR) 2025-02-19 EP disclosed
WO-2023198907-A1 SUBSTITUTED 6,7-DIHYDRO-5H-BENZO[7]ANNULENE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF SANOFI (FR) 2023-10-19 WO disclosed
US-8895582-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2014-11-25 US disclosed
US-8759374-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2014-06-24 US disclosed
US-20130053348-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS QIAN XIANGPING (US) 2013-02-28 US disclosed
US-20120135964-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS QIAN XIANGPING (US) 2012-05-31 US disclosed
US-20120022045-A1 BRIDGED COMPOUNDS AS HIV INTEGRASE INHIBITORS VENKATRAMAN SHANKAR (US) 2012-01-26 US disclosed
US-20120022045-A1 BRIDGED COMPOUNDS AS HIV INTEGRASE INHIBITORS VENKATRAMAN SHANKAR (US) 2012-01-26 US disclosed
EP-2391212-A1 BRIDGED COMPOUNDS AS HIV INTEGRASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2011-12-07 EP disclosed
US-8039507-B2 Therapeutic substituted gamma lactams ALLERGAN, INC. (US) 2011-10-18 US disclosed
WO-2010088167-A1 BRIDGED COMPOUNDS AS HIV INTEGRASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-08-05 WO disclosed
US-7705001-B2 Therapeutic substituted gamma lactams ALLERGAN, INC (US) 2010-04-27 US disclosed
US-20090239867-A1 THERAPEUTIC SUBSTITUTED GAMMA LACTAMS ALLERGAN, INC. (US) 2009-09-24 US disclosed
US-20080255220-A1 For treating inflammatory bowel disease, glaucoma or ocular hypertension, asthma; 7-[(3R*,4R*)-2-Oxo-4-((E)-3-oxo-oct-1-enyl)-pyrrolidin-3-yl]-hept-5-ynoic acid methyl ester; prostaglandin EP2 agonists ALLERGAN, INC. (US) 2008-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250263390-A1 NOVEL SUBSTITUTED 6,7-DIHYDRO-5H-BENZO[7]ANNULENE COMPOUNDS AND THEIR DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF GPER1, ESR2, ESRRA FKBP1A 1679/4885TOP2A 2334/4885DUT 4022/4885
US-20120022045-A1 BRIDGED COMPOUNDS AS HIV INTEGRASE INHIBITORS CCND3, CDK3, CDK2 FKBP1A 3582/4885TOP2A 123/4885DUT 264/4885
US-20090239867-A1 THERAPEUTIC SUBSTITUTED GAMMA LACTAMS DDO, DAO, GLA FKBP1A 1517/4885TOP2A 33/4885DUT 453/4885
US-20120135964-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS MYLK, MYH2, MYH10 FKBP1A 2736/4885TOP2A 262/4885DUT 2673/4885
US-20130053348-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS MYLK, MYH2, MYH10 FKBP1A 2736/4885TOP2A 262/4885DUT 2673/4885
US-20080255220-A1 For treating inflammatory bowel disease, glaucoma or ocular hypertension, asthma; 7-[(3R*,4R*)-2-Oxo-4-((E)-3-oxo-oct-1-enyl)-pyrrolidin-3-yl]-hept-5-ynoic acid methyl ester; prostaglandin EP2 agonists PTGIR, PTGIS, PTGER1 FKBP1A 1366/4885TOP2A 654/4885DUT 2299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.