SCHEMBL4225596

SCHEMBL4225596

CC(C)Nc1nc(-n2ccc(C(=O)O)n2)nc(Cl)c1-c1ccccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.35
MEN1 O00255 1/20 0.35
MAT2A P31153 2/20 0.34
GRM5 P41594 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MME P08473 1/20 0.32
MMEL1 Q495T6 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
LDHA P00338 1/20 0.31
LDHB P07195 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4231053 0.87 CXCL8 (0.32) KMT2AMAT2AGRM5CNR1CNR2
SCHEMBL4225599 0.85 MAT2A (0.33) MAT2ACNR1CNR2TSHRHTT
SCHEMBL4219849 0.82 KMT2A (0.45) KMT2AMEN1CNR1CNR2TSHR
SCHEMBL4232907 0.76 EGLN1 (0.40) CNR1CNR2LDHALDHB
SCHEMBL4219852 0.74 LMNA (0.35) KMT2AMEN1MAT2ACNR1CNR2
SCHEMBL4232192 0.72 EGLN1 (0.37) TSHRCYP2C19LDHALDHB
SCHEMBL4229598 0.71 KDM4E (0.34) KMT2AMEN1CNR1CNR2ALDH1A1
SCHEMBL4231674 0.69 LMNA (0.39) KMT2AMEN1CNR1CNR2TSHR
SCHEMBL4219785 0.69 GLP1R (0.42) KMT2AMEN1MAT2ACNR1CNR2
SCHEMBL4225977 0.68 HSP90AA1 (0.45) KMT2AMEN1CNR1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2092824-A1 Heterocyclyl pyrimidines Bayer CropScience AG (DE) 2009-08-26 EP disclosed