Betaprodine

Betaprodine

SCHEMBL4283575

CCC(=O)O[C@]1(c2ccccc2)CCN(C)C[C@@H]1C.c1ccc(C2(N3CCCCC3)CCCCC2)cc1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.77
DRD3 P35462 1/20 0.56
NPSR1 Q6W5P4 1/20 0.49
GRIN2D O15399 1/20 0.48
GRIN3B O60391 1/20 0.48
CYP2B6 P20813 1/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
PRCP P42785 1/20 0.48
SLC6A3 Q01959 1/20 0.48
GRIN1 Q05586 1/20 0.48
KCNH2 Q12809 1/20 0.48
GRIN2A Q12879 1/20 0.48
GRIN2B Q13224 1/20 0.48
GRIN2C Q14957 1/20 0.48
GRIN3A Q8TCU5 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
OPRM1 P35372 5/20 0.47
OPRD1 P41143 5/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Betaprodine SCHEMBL248367 0.88 LMNA (0.97) LMNADRD3NPSR1SLC6A4KCNH2
Betaprodine SCHEMBL186644 0.88 LMNA (0.97) LMNADRD3NPSR1SLC6A4KCNH2
Betaprodine SCHEMBL25053 0.88 LMNA (0.97) LMNADRD3NPSR1SLC6A4KCNH2
Alphaprodine SCHEMBL25054 0.88 LMNA (0.97) LMNADRD3NPSR1SLC6A4KCNH2
Alphaprodine SCHEMBL8818643 0.87 LMNA (1.00) LMNADRD3NPSR1SLC6A4KCNH2
Betaprodine SCHEMBL394431 0.87 LMNA (1.00) LMNADRD3NPSR1SLC6A4KCNH2
Betaprodine SCHEMBL1649307 0.86 LMNA (0.93) LMNADRD3NPSR1SLC6A4KCNH2
Proheptazine SCHEMBL25539 0.84 LMNA (0.84) LMNADRD3NPSR1SLC6A4KCNH2
SCHEMBL11541985 0.80 LMNA (0.70) LMNADRD3NPSR1SLC6A4KCNH2
SCHEMBL11383571 0.78 LMNA (0.78) LMNADRD3NPSR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9421266-B2 Safety of pseudoephedrine drug products PISGAH LABORATORIES, INC. (US) 2016-08-23 US disclosed
US-8859622-B1 Salts of physiologically active and psychoactive alkaloids and amines simultaneously exhibiting bioavailability and abuse resistance PISGAH LABORATORIES, INC. (US) 2014-10-14 US disclosed
US-20140178480-A1 SAFETY OF PSUEDOEPHEDRINE DRUG PRODUCTS PISGAH LABORATORIES, INC. 2014-06-26 US disclosed
US-8575151-B1 Salts of physiologically active and psychoactive alkaloids and amines simultaneously exhibiting bioavailability and abuse resistance Pisgah National Laboratories, Inc. (US) 2013-11-05 US disclosed
US-8334322-B1 Salts of physiologically active and psychoactive alkaloids and amines simultaneously exhibiting bioavailability and abuse resistance Pisgah Laboratories, LLC (US) 2012-12-18 US disclosed
US-20090259039-A1 Salts of physiologically active and psychoactive alkaloids and amines simultaneously exhibiting bioavailability and abuse resistance PISGAH LABORATORIES, INC. 2009-10-15 US disclosed
US-20080293695-A1 Salts of physiologically active and psychoactive alkaloids and amines simultaneously exhibiting bioavailability and abuse resistance PISGAH LABORATORIES, INC. 2008-11-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080293695-A1 Salts of physiologically active and psychoactive alkaloids and amines simultaneously exhibiting bioavailability and abuse resistance SLC6A2, SLC18A2, SLC6A3 LMNA 4559/4885DRD3 183/4885NPSR1 155/4885
US-20140178480-A1 SAFETY OF PSUEDOEPHEDRINE DRUG PRODUCTS SORD, ABCB11, ABCB1 LMNA 2816/4885DRD3 305/4885NPSR1 539/4885
US-20090259039-A1 Salts of physiologically active and psychoactive alkaloids and amines simultaneously exhibiting bioavailability and abuse resistance SLC18A2, SLC18A1, SLC6A2 LMNA 4054/4885DRD3 148/4885NPSR1 97/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.