Maleic Acid

Maleic Acid

SCHEMBL4301221

O=C(O)/C=C\C(=O)O.c1ccc(CCc2ccccc2)cc1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A known ✓ P35348 1/20 0.52
SLC6A3 known ✓ Q01959 1/20 0.52
ALDH1A1 P00352 5/20 0.66
TAAR1 Q96RJ0 3/20 0.66
HCAR2 Q8TDS4 3/20 0.66
LMNA P02545 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C19 P33261 1/20 0.59
FFAR1 O14842 1/20 0.58
KEAP1 Q14145 1/20 0.56
HDAC1 Q13547 4/20 0.52
HDAC3 O15379 2/20 0.52
HDAC4 P56524 2/20 0.52
HDAC7 Q8WUI4 2/20 0.52
HDAC2 Q92769 2/20 0.52
HDAC10 Q969S8 2/20 0.52
HDAC11 Q96DB2 2/20 0.52
HDAC8 Q9BY41 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
HDAC9 Q9UKV0 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL4074902 0.93 ALDH1A1 (0.59) ALDH1A1TAAR1HCAR2LMNACYP2D6
Cinnamic Acid SCHEMBL890441 0.85 HCAR2 (0.76) ALDH1A1HCAR2LMNACYP2D6CYP2C19
SCHEMBL23854259 0.83 HDAC3 (0.67) HCAR2FFAR1HDAC1HDAC3HDAC4
SCHEMBL3225302 0.83 HDAC3 (0.67) HCAR2FFAR1HDAC1HDAC3HDAC4
Butylbenzyl SCHEMBL28319138 0.83 ATG4B (0.63) ALDH1A1TAAR1HCAR2TDP1
SCHEMBL2856224 0.82 GPR52 (0.70) GPR52
SCHEMBL2853640 0.82 GPR52 (0.70) GPR52
SCHEMBL2853636 0.82 GPR52 (0.70) GPR52
Phenylacetic Acid SCHEMBL30960397 0.81 AKR1B1 (0.77) ALDH1A1TAAR1HCAR2LMNACYP2D6
Benzylamine SCHEMBL8533927 0.81 LOXL2 (0.64) ALDH1A1TAAR1HCAR2LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153737-A The manufacturing method of terminal-modified conjugated diolefin polymer, rubber composition, rubber product and terminal-modified conjugated diolefin polymer 株式会社普利司通 2019-01-04 CN disclosed
CN-103044921-B Photo curable organopolysiloxane composition 信越化学工业株式会社 2017-03-01 CN disclosed
US-20090267489-A1 GAS BARRIER THIN FILM LAMINATE, GAS BARRIER RESIN SUBSTRATE AND ORGANIC EL DEVICE KONICA MINOLTA HOLDINGS, INC. (JP) 2009-10-29 US disclosed