SCHEMBL4316404

SCHEMBL4316404

Cn1cnc2c1c(=O)n(CC(=O)[O-])c(=O)n2C.[Na+]

nearest known ligand 0.75

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B known ✓ P29275 8/20 0.75
PDE4A known ✓ P27815 1/20 0.61
PDE4B known ✓ Q07343 1/20 0.61
PDE4C known ✓ Q08493 1/20 0.61
PDE4D known ✓ Q08499 1/20 0.61
ADORA3 known ✓ P0DMS8 1/20 0.56
ADORA2A known ✓ P29274 1/20 0.56
ADORA1 known ✓ P30542 1/20 0.56
TNF P01375 4/20 0.61
ACHE P22303 2/20 0.61
USP2 O75604 1/20 0.61
LMNA P02545 1/20 0.61
CYP1A2 P05177 1/20 0.61
TSHR P16473 1/20 0.61
NFKB1 P19838 1/20 0.61
PMP22 Q01453 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
RXFP1 Q9HBX9 1/20 0.61
GLA P06280 1/20 0.59
BLM P54132 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Zinc Ion SCHEMBL10408407 0.97 ADORA2B (0.75) ADORA2BTNFACHEUSP2LMNA
SCHEMBL10407485 0.97 ADORA2B (0.75) ADORA2BTNFACHEUSP2LMNA
SCHEMBL10407724 0.97 ADORA2B (0.75) ADORA2BTNFACHEUSP2LMNA
SCHEMBL10407732 0.97 ADORA2B (0.75) ADORA2BTNFACHEUSP2LMNA
SCHEMBL10407721 0.86 PDE4A (0.63) ADORA2BTNFACHEUSP2LMNA
SCHEMBL10407729 0.86 PDE4A (0.63) ADORA2BTNFACHEUSP2LMNA
SCHEMBL10407483 0.86 PDE4A (0.63) ADORA2BTNFACHEUSP2LMNA
Zinc Ion SCHEMBL10408405 0.86 PDE4A (0.63) ADORA2BTNFACHEUSP2LMNA
SCHEMBL20863739 0.86 ADORA2B (1.00) ADORA2BTNFACHEUSP2LMNA
SCHEMBL356160 0.86 ADORA2B (1.00) ADORA2BTNFACHEUSP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111110590-B Agar oligosaccharide composition for balancing scalp grease secretion, preparation method and application 厦门传茗生物科技有限公司 2022-06-28 CN disclosed
US-10877035-B2 Advanced drug development and manufacturing ICAGEN, LLC (US) 2020-12-29 US disclosed
CN-111110590-A Agar oligosaccharide composition for balancing scalp grease secretion, preparation method and application 蓝脑科技(厦门)有限公司 2020-05-08 CN disclosed
US-20150309021-A1 Advanced Drug Development and Manufacturing LOS ALAMOS NATIONAL SECURITY, LLC 2015-10-29 US disclosed
EP-2511844-B1 X-ray microscope XRPRO SCIENCES INC (US) 2015-08-12 EP disclosed
EP-2511844-A2 Advanced drug development and manufacturing Los Alamos National Security, LLC (US) 2012-10-17 EP disclosed
EP-2084519-B1 X-RAY FLUORESCENCE ANALYSIS METHOD LOS ALAMOS NAT SECURITY LLC (US) 2012-08-01 EP disclosed
EP-2084519-A2 ADVANCED DRUG DEVELOPMENT AND MANUFACTURING Los Alamos National Security, LLC (US) 2009-08-05 EP disclosed
WO-2008127291-A2 ADVANCED DRUG DEVELOPMENT AND MANUFACTURING LOS ALAMOS NATIONAL SECURITY, LLC (US) 2008-10-23 WO disclosed
US-20080220441-A1 Advanced drug development and manufacturing THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2008-09-11 US disclosed