SCHEMBL4336775

SCHEMBL4336775

CC(C)O[C@@H](CC(=O)O)c1cccc(CNC(=O)OCc2ccnc3ccccc23)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.41
NSD2 O96028 1/20 0.41
TNKS O95271 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
DNMT1 P26358 1/20 0.39
DNMT3A Q9Y6K1 1/20 0.39
CASP1 P29466 3/20 0.39
CASP3 P42574 1/20 0.38
ADAMTS4 O75173 1/20 0.37
MMP13 P45452 1/20 0.37
KCNA5 P22460 1/20 0.37
NAMPT P43490 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
ADAM17 P78536 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4336772 0.83 EPHX1 (0.42) EPHX1NSD2TNKSTNKS2DNMT1
SCHEMBL4336778 0.83 EPHX1 (0.42) EPHX1NSD2TNKSTNKS2DNMT1
SCHEMBL4329711 0.82 CYSLTR1 (0.49)
SCHEMBL4334154 0.80 LMNA (0.44) CASP1ALDH1A1MAPT
SCHEMBL4339537 0.80 HDAC1 (0.40) EPHX1TNKSTNKS2KCNA5NAMPT
SCHEMBL4342514 0.79 ALDH1A1 (0.42) CASP3ALDH1A1MAPT
SCHEMBL4348232 0.79 CASP1 (0.36) EPHX1TNKSTNKS2CASP1CASP3
SCHEMBL4334667 0.78 NPC1 (0.49) CASP1ALDH1A1MAPT
SCHEMBL4334187 0.78 FFAR1 (0.49)
SCHEMBL4337917 0.77 NR3C2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7544835-B2 Carboxylic acid derivative and salt thereof EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-06-09 US disclosed