SCHEMBL434387

SCHEMBL434387

O=C(O)c1cccc(C2(C(=O)N(CCN3CCCC3)c3ccccc3)CC2)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HIF1A Q16665 1/20 0.43
PTGIR P43119 1/20 0.41
KMT2A Q03164 5/20 0.41
MEN1 O00255 2/20 0.41
OPRM1 P35372 3/20 0.40
GAA P10253 2/20 0.40
MAPK1 P28482 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
ALDH1A1 P00352 5/20 0.40
GFER P55789 1/20 0.39
KDM4E B2RXH2 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HSD11B1 P28845 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433443 0.92 HRH3 (0.43) HRH3PTGIRKMT2AMEN1OPRM1
SCHEMBL434778 0.77 PTGIR (0.44) HRH3PTGIRKMT2AMEN1GAA
SCHEMBL4931908 0.69 HRH3 (0.53) HRH3PTGIRKMT2AOPRM1SIGMAR1
SCHEMBL8437918 0.69 OPRM1 (0.51) HRH3PTGIRKMT2AOPRM1SIGMAR1
SCHEMBL15380628 0.69 ALDH1A1 (0.44) CYP2D6CYP2C9HIF1AKMT2AMEN1
SCHEMBL432280 0.69 ALDH1A1 (0.44) CYP2D6CYP2C9HIF1AKMT2AMEN1
SCHEMBL6209135 0.67 PDK1 (0.47) HRH3PTGIRKMT2AOPRM1SIGMAR1
SCHEMBL5758121 0.66 ADRA2C (0.61) PTGIRKMT2AALDH1A1GFERKDM4E
SCHEMBL4233535 0.66 PDK1 (0.49) HRH3PTGIRKMT2AOPRM1SIGMAR1
Hydrochloric Acid SCHEMBL5071191 0.66 PDK1 (0.47) HRH3PTGIRKMT2AMEN1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO claimed