SCHEMBL435603

SCHEMBL435603

Fc1cc[c]c(-c2ccc(Cl)cc2F)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.35
EGLN2 Q96KS0 1/20 0.34
GRM2 Q14416 4/20 0.32
HSD11B1 P28845 1/20 0.32
PSEN1 P49768 4/20 0.32
PSEN2 P49810 4/20 0.32
APH1B Q8WW43 4/20 0.32
NCSTN Q92542 4/20 0.32
APH1A Q96BI3 4/20 0.32
PSENEN Q9NZ42 4/20 0.32
S100A4 P26447 1/20 0.31
CNR1 P21554 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31
CLK1 P49759 1/20 0.31
PTGS2 P35354 1/20 0.31
GPR3 P46089 1/20 0.31
CCR2 P41597 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433550 0.89 KMO (0.36) KMOEGLN2GRM2HSD11B1S100A4
SCHEMBL435140 0.86 AHR (0.40) HSD11B1
SCHEMBL434555 0.86 CNR1 (0.34) KMOCNR1TAS1R3TAS1R1TAS1R2
SCHEMBL433493 0.85 ALDH1A1 (0.37) KMOPTGS2GPR3
SCHEMBL9648679 0.79 L3MBTL1 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9139645 0.79 EGLN2 (0.37) KMOEGLN2
SCHEMBL434680 0.79 GPR3 (0.38) KMOEGLN2GRM2HSD11B1S100A4
SCHEMBL6927659 0.78 NISCH (0.40) GRM2HSD11B1CLK1PTGS2
SCHEMBL2053480 0.76 CA3 (0.33) TAS1R3TAS1R1TAS1R2
SCHEMBL434431 0.76 L3MBTL1 (0.38) GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016026830-A1 NOVEL FUNGICIDAL PYRAZOLE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-25 WO disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed