SCHEMBL441951

SCHEMBL441951

Nc1c(Br)cnc2c(Cl)cccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.58
NR4A2 P43354 3/20 0.51
ACHE P22303 2/20 0.44
AURKA O14965 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
PRKD3 O94806 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
ABL1 P00519 1/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41
IGF1R P08069 1/20 0.41
MET P08581 1/20 0.41
PDGFRB P09619 1/20 0.41
PARP1 P09874 1/20 0.41
PIM1 P11309 1/20 0.41
FGFR1 P11362 1/20 0.41
PDGFRA P16234 1/20 0.41
PRKACA P17612 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL441707 0.83 HAVCR2 (0.63) HAVCR2NR4A2ACHEAURKADAPK3
SCHEMBL442133 0.83 BACE1 (0.41) HAVCR2NR4A2FGFR1GSK3BCDK5
SCHEMBL441701 0.79 ALDH1A1 (0.43) HAVCR2PARP1CYP1A2CYP2A6LMNA
SCHEMBL435823 0.79 PARP1 (0.41) HAVCR2PARP1CYP1A2ALDH1A1MEN1
SCHEMBL439423 0.79 HAVCR2 (0.36) HAVCR2LMNAALDH1A1MEN1MAPT
SCHEMBL437767 0.79 HAVCR2 (0.46) HAVCR2NR4A2ACHECHEK1FLT3
SCHEMBL440009 0.76 HAVCR2 (0.38) HAVCR2ALDH1A1MEN1MAPTKMT2A
SCHEMBL438876 0.75 BCHE (0.43) HAVCR2ACHEDYRK1AALDH1A1MAPT
SCHEMBL440370 0.75 PARP1 (0.45) PRKD3MAP4K4PARP1CLK2GSK3A
SCHEMBL435849 0.75 HTR1A (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed