SCHEMBL4361885

SCHEMBL4361885

CS(=O)(=O)c1nccc(Oc2ccc(N)c(N)c2)n1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.43
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDR P35968 16/20 0.36
RET P07949 2/20 0.33
FLT1 P17948 2/20 0.33
IKBKB O14920 1/20 0.32
MET P08581 1/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28281419 0.78 PGR (0.44) LMNASMN1; SMN2
SCHEMBL6972835 0.78 SDHB (0.40) LMNASMN1; SMN2KDRMET
SCHEMBL4364798 0.76 ALDH1A1 (0.50) LMNASMN1; SMN2IKBKB
SCHEMBL4367250 0.74 HTT (0.56) NR4A1LMNASMN1; SMN2KDR
SCHEMBL4363839 0.74 NR4A1 (0.46) NR4A1KDRMET
SCHEMBL8669831 0.74 ALDH1A1 (0.53) LMNAKDRRETFLT1PDGFRB
SCHEMBL7270618 0.72 SMN1; SMN2 (0.60) LMNASMN1; SMN2
SCHEMBL32665306 0.71 LMNA (0.42) LMNASMN1; SMN2
SCHEMBL2261767 0.69 SMN1; SMN2 (0.38) LMNASMN1; SMN2
SCHEMBL2411422 0.69 SMN1; SMN2 (0.43) LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed
EP-1638954-A1 FUSED AZOLES SUCH AS 2,5-DISUBSTITUTED BENZIMIDAZOLES, BENZOXAZOLES AND BENZOTHIAZOLES AS KINASE INHIBITORS AMGEN INC. (US) 2006-03-29 EP disclosed
US-20040209892-A1 Heterocyclic compounds and methods of use U.S. PATENT OPERATIONS 2004-10-21 US disclosed
WO-2004085425-A1 FUSED AZOLES SUCH AS 2,5-DISUBSTITUTED BENZIMIDAZOLES, BENZOXAZOLES AND BENZOTHIAZOLES AS KINASE INHIBITORS AMGEN INC (US) 2004-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209892-A1 Heterocyclic compounds and methods of use VHL, NQO1, HPGDS NR4A1 2382/4885LMNA 2395/4885SMN1; SMN2 2240/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.