Safrazine

Safrazine

SCHEMBL437129

CC(CCc1ccc2c(c1)OCO2)NN

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.57
SLC6A4 P31645 3/20 0.57
SLC6A2 P23975 2/20 0.57
SLC6A3 Q01959 2/20 0.57
CYP2D6 P10635 1/20 0.57
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
TSHR P16473 1/20 0.56
ADRB2 P07550 3/20 0.50
ADRB1 P08588 3/20 0.50
ADRB3 P13945 3/20 0.50
ADRA1D P25100 2/20 0.50
ADRA1A P35348 2/20 0.50
ADRA1B P35368 2/20 0.50
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
POLB P06746 1/20 0.49
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Safrazine SCHEMBL29359452 1.00 TAAR1 (0.57) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
Safrazine SCHEMBL1868031 0.98 TAAR1 (0.56) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL10395528 0.84 TAAR1 (0.74) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL987525 0.83 TAAR1 (0.71) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL8294114 0.82 TAAR1 (0.61) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL31303188 0.80 TAS1R3 (0.55) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL2485767 0.80 TAAR1 (0.57) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL29664514 0.80 TAAR1 (0.57) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL28123545 0.80 TAAR1 (0.57) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL10715342 0.79 ALDH1A1 (0.64) TAAR1SLC6A4SLC6A2SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 496 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260001942-A1 TREATMENT OF HEADACHE DISORDERS AND/OR PSYCHIATRIC SYMPTOMS USING ANTI-CGRP ANTIBODIES, AND COMPOSITIONS AND METHODS RELATED THERETO H LUNDBECK AS (DK) 2026-01-01 US claimed
WO-2025262247-A1 TREATMENT OF HEADACHE DISORDERS AND/OR PSYCHIATRIC SYMPTOMS USING ANTI-CGRP ANTIBODIES, AND COMPOSITIONS AND METHODS RELATED THERETO H. LUNDBECK A/S (DK) 2025-12-26 WO claimed
US-20250339403-A1 Tryptamine Formulations and Uses Thereof Natural MedTech Pty Ltd (AU) 2025-11-06 US claimed
EP-4618981-A1 COMBINATIONS OF MONOAMINE OXIDASE INHIBITORS AND SEROTONIN RECEPTOR AGONISTS AND THEIR THERAPEUTIC USE Remedi, Inc. (US) 2025-09-24 EP claimed
EP-4615444-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural Medtech Pty Ltd (AU) 2025-09-17 EP claimed
WO-2025151884-A1 USE OF GLYCOSAMINOGLYCAN SULFATED POLYSACCHARIDES SUCH AS SODIUM PENTOSAN POLYSULFATE IN COMBINATION WITH PERMEATION AGENTS TO TREAT ALZHEIMER'S DISEASE PARSONS C LOWELL (US) 2025-07-17 WO claimed
EP-4479032-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS Sage Therapeutics, Inc. (US) 2024-12-25 EP claimed
US-12121513-B2 Betahistine, or a pharmaceutically acceptable salt thereof, and a monoamine oxidase inhibitor, for use in the treatment or prevention of one or more symptoms of vertigo in a subject Intrabio Ltd. (GB) 2024-10-22 US claimed
WO-2024108195-A1 COMBINATIONS OF MONOAMINE OXIDASE INHIBITORS AND SEROTONIN RECEPTOR AGONISTS AND THEIR THERAPEUTIC USE REMEDI, INC. (US) 2024-05-23 WO claimed
WO-2024098098-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural MedTech Pty Ltd (AU) 2024-05-16 WO claimed
EP-1991248-A2 ANTIDEPRESSANT PRODRUGS Shire LLC (US) 2008-11-19 EP claimed
WO-2007100668-A2 ANTIDEPRESSANT PRODRUGS SHIRE LLC (US) 2007-09-07 WO claimed
US-20060287299-A1 Combination therapy for dementia, depression and apathy SHELDON LESLIE J 2006-12-21 US claimed
EP-1713486-A1 COMBINATION THERAPY FOR DEMENTIA,DEPRESSION AND APATHY Sheldon, Leslie James (CA) 2006-10-25 EP claimed
US-6946141-B2 As-needed administration of tricyclic and other non-SRI antidepressant drugs to treat premature ejaculation VIVUS, INC. (US) 2005-09-20 US claimed
WO-2005053703-A1 COMBINATION THERAPY FOR DEMENTIA, DEPRESSION AND APATHY SHELDON LESLIE JAMES (CA) 2005-06-16 WO claimed
WO-2004041207-A2 GHB TREATMENT METHODS BAYLOR RESEARCH INSTITUTE (US) 2004-05-21 WO claimed
EP-1389115-A2 AS-NEEDED ADMINISTRATION OF TRICYCLIC AND OTHER NON-SRI ANTIDEPRESSANT DRUGS TO TREAT PREMATURE EJACULATION Vivus, Inc. (US) 2004-02-18 EP claimed
US-20020161016-A1 As-needed administration of tricyclic and other non-SRI antidepressant drugs to treat premature ejaculation VIVUS LLC (F/K/A VIVUS, INC.) 2002-10-31 US claimed
WO-2002041883-A2 AS-NEEDED ADMINISTRATION OF TRICYCLIC AND OTHER NON-SRI ANTIDEPRESSANT DRUGS TO TREAT PREMATURE EJACULATION VIVUS, INC. (US) 2002-05-30 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020161016-A1 As-needed administration of tricyclic and other non-SRI antidepressant drugs to treat premature ejaculation HTR5A, HTR1A, MAOA TAAR1 150/4885SLC6A4 214/4885SLC6A2 160/4885
US-20260001942-A1 TREATMENT OF HEADACHE DISORDERS AND/OR PSYCHIATRIC SYMPTOMS USING ANTI-CGRP ANTIBODIES, AND COMPOSITIONS AND METHODS RELATED THERETO CDR2, OPRL1, TPH1 TAAR1 350/4885SLC6A4 221/4885SLC6A2 314/4885
US-12121513-B2 Betahistine, or a pharmaceutically acceptable salt thereof, and a monoamine oxidase inhibitor, for use in the treatment or prevention of one or more symptoms of vertigo in a subject HNMT, MAOA, MAOB TAAR1 655/4885SLC6A4 73/4885SLC6A2 6/4885
US-20250339403-A1 Tryptamine Formulations and Uses Thereof MAOA, MAOB, TPH1 TAAR1 55/4885SLC6A4 36/4885SLC6A2 28/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.