Toluene

Toluene

SCHEMBL437383

Cc1ccccc1.Cc1ccccc1.Cc1ccccc1.Cc1ccccc1.O=P(O)(O)O.O=P(O)(O)O

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Toluene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.65
TSHR P16473 2/20 0.65
ALOX12 P18054 1/20 0.65
ACHE P22303 1/20 0.65
ACP3 P15309 2/20 0.50
CA2 P00918 1/20 0.50
CA4 P22748 1/20 0.50
CA5A P35218 1/20 0.50
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
MAPT P10636 1/20 0.45
SRC P12931 2/20 0.44
CFTR P13569 1/20 0.44
POLB P06746 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PTPN1 P18031 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Toluene SCHEMBL5806354 1.00 LMNA (0.65) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL10856877 1.00 LMNA (0.65) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL28555681 1.00 LMNA (0.65) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL695755 1.00 LMNA (0.65) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL27269290 1.00 LMNA (0.65) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL1011089 1.00 LMNA (0.65) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL1931900 0.97 LMNA (0.61) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL3630619 0.97 LMNA (0.61) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL27955550 0.97 LMNA (0.61) LMNATSHRALOX12ACHEACP3
Toluene SCHEMBL29009365 0.97 LMNA (0.61) LMNATSHRALOX12ACHEACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 141 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11298367-B2 Prodrugs of substituted triazole derivatives and uses thereof BAYER AKTIENGESELLSCHAFT (DE) 2022-04-12 US claimed
EP-3700913-B1 PRODRUGS OF SUBSTITUTED TRIAZOLE DERIVATIVES AND USES THEREOF BAYER AG (DE) 2021-11-10 EP claimed
US-20200338096-A1 PRODRUGS OF SUBSTITUTED TRIAZOLE DERIVATIVES AND USES THEREOF BAYER AKTIENGESELLSCHAFT (DE) 2020-10-29 US claimed
EP-3700913-A1 PRODRUGS OF SUBSTITUTED TRIAZOLE DERIVATIVES AND USES THEREOF Bayer Aktiengesellschaft (DE) 2020-09-02 EP claimed
CN-111225921-A Prodrugs of substituted triazole derivatives and uses thereof 拜耳股份公司 2020-06-02 CN claimed
US-20260097111-A1 ETHER LIPIDS FOR HYPERACTIVATION OF MAMMALIAN DENDRITIC CELLS CORNER THERAPEUTICS, INC. (US) 2026-04-09 US disclosed
EP-4720063-A1 NAPHTHYRIDINONE DERIVATIVES FOR THE TREATMENT OF A DISEASE OR DISORDER Novartis AG (CH) 2026-04-08 EP disclosed
EP-4714961-A2 PRODRUG MODULATORS OF THE INTEGRATED STRESS PATHWAY Calico Life Sciences LLC (US) 2026-03-25 EP disclosed
EP-4209483-B1 PRODRUG MODULATORS OF THE INTEGRATED STRESS PATHWAY CALICO LIFE SCIENCES LLC (US) 2025-12-03 EP disclosed
US-12421276-B2 Methods of treating neurodegenerative disease with substituted n-hexanoic-l-tyrosine-l-isoleucine-(6)-aminohexanoic amide analogues ATHIRA PHARMA, INC. (US) 2025-09-23 US disclosed
US-20250275991-A1 ORAL COMPLEMENT FACTOR D INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2025-09-04 US disclosed
EP-4604919-A1 ETHER LIPIDS FOR HYPERACTIVATION OF MAMMALIAN DENDRITIC CELLS Corner Therapeutics, Inc. (US) 2025-08-27 EP disclosed
US-20100221269-A1 SYNTHETIC LIPID A DERIVATIVE UNIVERSITY OF GEORGIA RESEACH FOUNDATION, INC (US) 2010-09-02 US disclosed
WO-2010047737-A2 ANTIMICROBIAL INDOLINE COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. (KY) 2010-04-29 WO disclosed
US-20100069441-A1 ANTIMICROBIAL INDOLINE COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS GORDEEV MIKHAIL FEDOROVICH 2010-03-18 US disclosed
WO-2009035528-A2 SYNTHETIC LIPID A DERIVATIVE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2009-03-19 WO disclosed
EP-1283672-B1 ANTITUBULIN ASSEMBLY AND CELL GROWTH INHIBITOR DENOMINATED \"DIOXOSTATIN\ UNIV ARIZONA STATE (US) 2004-11-17 EP disclosed
US-20040122083-A1 Antitubulin assembly and cell growth inhibitor denominated \"dioxostatin\ ARIZONA BOARD OF REGENTS ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY 2004-06-24 US disclosed
EP-1283672-A1 ANTITUBULIN ASSEMBLY AND CELL GROWTH INHIBITOR DENOMINATED \"DIOXOSTATIN\ Arizona Board of Regents, acting for and on behalf of Arizona State University (US) 2003-02-19 EP disclosed
WO-2001084929-A1 ANTITUBULIN ASSEMBLY AND CELL GROWTH INHIBITOR DENOMINATED 'DIOXOSTATIN' ARIZONA BOARD OF REGENTS, ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2001-11-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200338096-A1 PRODRUGS OF SUBSTITUTED TRIAZOLE DERIVATIVES AND USES THEREOF CYP4B1, AADAC, GLS LMNA 1534/4885TSHR 1793/4885ALOX12 3571/4885
US-20250275991-A1 ORAL COMPLEMENT FACTOR D INHIBITORS CFD, CFH, CFB LMNA 1900/4885TSHR 3081/4885ALOX12 423/4885
US-20040122083-A1 Antitubulin assembly and cell growth inhibitor denominated \"dioxostatin\ MCL1, TUBA1C, TUBB8 LMNA 2780/4885TSHR 2903/4885ALOX12 4699/4885
US-20100069441-A1 ANTIMICROBIAL INDOLINE COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS IDO1, IDO2, INMT LMNA 2380/4885TSHR 4027/4885ALOX12 2647/4885
US-20260097111-A1 ETHER LIPIDS FOR HYPERACTIVATION OF MAMMALIAN DENDRITIC CELLS TLR7, INPP5D, PLCD1 LMNA 3757/4885TSHR 951/4885ALOX12 1241/4885
US-12421276-B2 Methods of treating neurodegenerative disease with substituted n-hexanoic-l-tyrosine-l-isoleucine-(6)-aminohexanoic amide analogues AADAT, ABAT, IAPP LMNA 2873/4885TSHR 2069/4885ALOX12 616/4885
US-20100221269-A1 SYNTHETIC LIPID A DERIVATIVE DDOST, STT3A, UGCG LMNA 2345/4885TSHR 1943/4885ALOX12 495/4885
US-11298367-B2 Prodrugs of substituted triazole derivatives and uses thereof CYP4B1, AADAC, GLS LMNA 1534/4885TSHR 1793/4885ALOX12 3571/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.