SCHEMBL4374417

SCHEMBL4374417

CC(C)(C)C(NC(=O)O)C(N)c1ccccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
CYP2D6 P10635 1/20 0.40
NFKB1 P19838 1/20 0.40
HIF1A Q16665 1/20 0.40
BLM P54132 1/20 0.39
CTSA P10619 3/20 0.38
AOC3 Q16853 1/20 0.38
KMT2A Q03164 1/20 0.37
CXCL8 P10145 3/20 0.37
PRSS1 P07477 1/20 0.36
CTSG P08311 1/20 0.36
CTRB1 P17538 1/20 0.36
CMA1 P23946 1/20 0.36
CASP1 P29466 1/20 0.36
SLC1A3 P43003 1/20 0.36
SLC1A2 P43004 1/20 0.36
SLC1A1 P43005 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ACP3 P15309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4584586 0.82 GAA (0.46) HIF1ACTSAKMT2A
SCHEMBL4387389 0.80 CNR2 (0.46) CTSAACP3
SCHEMBL4371317 0.80 ALDH1A1 (0.48)
SCHEMBL4377187 0.80 DPP4 (0.43) KMT2ACTRB1L3MBTL1
SCHEMBL4373941 0.80 DPP4 (0.43) KMT2ACTRB1L3MBTL1
SCHEMBL4380602 0.76 PRCP (0.41) ADRB2CYP2D6NFKB1BLMKMT2A
SCHEMBL4371128 0.74 TRPM8 (0.41) BLMKMT2AACP3
SCHEMBL11244690 0.73 CXCL8 (0.44) ADRB2ADRB1HIF1ACTSAAOC3
SCHEMBL4596289 0.71 ADRB2 (0.51) ADRB2ADRB1CYP2D6NFKB1HIF1A
SCHEMBL4584032 0.71 HDAC4 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117523-A1 INHIBITORS OF AKT ACTIVITY SmithKline Beecham Corporation (US) 2009-11-18 EP disclosed
WO-2008098104-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-08-14 WO disclosed