SCHEMBL4386498

SCHEMBL4386498

O=C(NC1CCCCn2c1nc(-c1ccncc1)cc2=O)c1cccnc1Sc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
ATM Q13315 1/20 0.41
CGAS Q8N884 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 3/20 0.38
P2RX7 Q99572 1/20 0.37
CYP2C9 P11712 3/20 0.37
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD11B1 P28845 1/20 0.36
CNR1 P21554 2/20 0.35
CNR2 P34972 2/20 0.35
CDC7 O00311 1/20 0.35
MAP4K4 O95819 1/20 0.35
PIM1 P11309 1/20 0.35
PRKACA P17612 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4377829 0.93 ALDH1A1 (0.45) ALDH1A1HTTSMN1; SMN2CGASRAB9A
SCHEMBL4385766 0.90 RAB9A (0.51) ALDH1A1HTTRAB9AKMT2ACYP2C9
SCHEMBL4948489 0.86 HSD11B1 (0.54) ALDH1A1HTTRAB9AKMT2AMEN1
SCHEMBL4391283 0.85 CYP2C9 (0.39) ALDH1A1CGASKMT2ACYP2C9MEN1
SCHEMBL4391863 0.85 MAPT (0.40) ALDH1A1SMN1; SMN2CGASRAB9AKMT2A
SCHEMBL4952879 0.84 MEN1 (0.47) ALDH1A1CGASKMT2ACYP2C9MEN1
SCHEMBL4383616 0.81 MEN1 (0.47) ALDH1A1KMT2AMEN1CNR1CNR2
SCHEMBL2065962 0.81 KMT2A (0.46) ALDH1A1CGASKMT2AMEN1GSK3B
SCHEMBL2066118 0.81 ALDH1A1 (0.43) ALDH1A1CGASRAB9AKMT2AMEN1
SCHEMBL4387186 0.80 L3MBTL1 (0.56) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP claimed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO claimed
EP-1939187-A1 Substituted heteroaryl pyridopyrimidone derivatives Sanofi-Aventis (FR) 2008-07-02 EP claimed
US-8198287-B2 Substituted heteroaryl pyridopyrimidone derivatives SANOFI-AVENTIS (FR) 2012-06-12 US disclosed
EP-1939187-A1 Substituted heteroaryl pyridopyrimidone derivatives Sanofi-Aventis (FR) 2008-07-02 EP disclosed