SCHEMBL4387383

SCHEMBL4387383

COc1ccc(-c2ccc(CN3CCNCC3=O)cc2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.45
TEK Q02763 4/20 0.45
NAAA Q02083 1/20 0.42
INSR P06213 1/20 0.42
ALK Q9UM73 1/20 0.42
EPHB4 P54760 3/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
PRMT5 O14744 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
CYP11B1 P15538 1/20 0.41
PDE1B Q01064 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
MRGPRX1 Q96LB2 1/20 0.40
CHEK1 O14757 1/20 0.40
PIK3CA P42336 1/20 0.40
MTOR P42345 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20133743 0.78 GAA (0.57)
SCHEMBL7996202 0.76 ENPP2 (0.51) ACHE
SCHEMBL24648953 0.73 MGLL (0.43) HTR2AHTR2CHTR2B
SCHEMBL18291305 0.73 CHRM1 (0.44) PRMT5
SCHEMBL18076484 0.72 GAA (0.53) ACHE
SCHEMBL3594508 0.72 CHRNB2 (0.56) CHRNB2CHRNA4
SCHEMBL4692001 0.72 MEN1 (0.47)
Hydrochloric Acid SCHEMBL1583990 0.71 CHRNB2 (0.54) CHRNB2CHRNA4
SCHEMBL14863940 0.70 HTR2C (0.43) HTR2C
SCHEMBL25271016 0.70 ALDH1A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612075-B2 Substituted oxoazaheterocyclyl compounds AVENTIS PHARMACEUTICALS INC. (US) 2009-11-03 US disclosed