SCHEMBL4394026

SCHEMBL4394026

O=CCCc1ccccc1S

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
GPR52 Q9Y2T5 1/20 0.31
FOLH1 Q04609 1/20 0.31
ADH1B P00325 1/20 0.30
ADH1C P00326 1/20 0.30
ADH1A P07327 1/20 0.30
ADH7 P40394 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28607303 0.84 ADH1B (0.36) GPR52FOLH1ADH1BADH1CADH1A
SCHEMBL28552014 0.78 TLR8 (0.37)
SCHEMBL5174795 0.78 IDO1 (0.36) MAPTHDAC8FOLH1
SCHEMBL1738495 0.77 MAPT (0.33) MAPTHDAC8
SCHEMBL910692 0.76 GABRA1 (0.39) MAPT
SCHEMBL8414772 0.76 MAPT (0.32) MAPTHDAC8
SCHEMBL143458 0.75 MTNR1A (0.49) MAPT
SCHEMBL587837 0.75 IDO1 (0.36) MAPTHDAC8
SCHEMBL4444470 0.74 LMNA (0.50)
SCHEMBL1338205 0.74 TAAR1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7574340-B2 Small molecules and a pharmacophore model for inhibition of botulinum toxin and methods of making and using thereof THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 2009-08-11 US disclosed
US-20050153945-A1 Small molecules and a pharmacophore model for inhibition of botulinum toxin and methods of making and using thereof ARMY, UNITED STATES 2005-07-14 US disclosed
WO-2005026193-A2 SMALL MOLECULES AND A PHARMACOPHORE MODEL FOR INHIBITION OF BOTULINUM TOXIN AND METHODS OF MAKING AND USING THEREOF UNITED STATES ARMY MEDICAL RESEARCH AND MATERIEL COMMAND (US) 2005-03-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050153945-A1 Small molecules and a pharmacophore model for inhibition of botulinum toxin and methods of making and using thereof MMP2, RAC2, RAC1 MAPT 4644/4885HDAC8 2856/4885GPR52 1237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.