SCHEMBL439770

SCHEMBL439770

Nc1c(Cl)cnc2ccc(C(F)(F)F)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.42
NPBWR1 P48145 2/20 0.41
EPHX2 P34913 1/20 0.41
SCN4A P35499 1/20 0.41
NOS3 P29474 1/20 0.40
NOS2 P35228 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
EGFR P00533 3/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 1/20 0.37
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
KDM1A O60341 1/20 0.36
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
DYRK3 O43781 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438632 0.87 PARP1 (0.45) BACE1NPBWR1NOS3NOS2ALDH1A1
SCHEMBL23935164 0.83 BACE1 (0.45) BACE1NPBWR1EPHX2SCN4ANOS3
SCHEMBL29742208 0.83 BACE1 (0.45) BACE1NPBWR1EPHX2SCN4ANOS3
SCHEMBL436530 0.81 BACE1 (0.42) BACE1NPBWR1EPHX2SCN4ANOS3
SCHEMBL439645 0.78 ACHE (0.46) BACE1CYP1A2MAP4K4AXL
SCHEMBL439464 0.78 NR4A2 (0.55) EGFRCYP1A2MAP4K4CYP2D6
SCHEMBL437175 0.77 NPC1 (0.44) SCN4ASMN1; SMN2CYP1A2CYP3A4CDK2
SCHEMBL439948 0.76 ALDH1A1 (0.53) ALDH1A1KDM4ECYP1A2CHEK1AURKA
SCHEMBL18658922 0.75 ALDH1A1 (0.47) BACE1ALDH1A1KDM4EPOLBCYP3A4
SCHEMBL30050271 0.75 CCNC (0.48) BACE1NOS3NOS2KDM4EEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed