SCHEMBL438632

SCHEMBL438632

Nc1c(Cl)cnc2cc(C(F)(F)F)ccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
MAOB P27338 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
NOS3 P29474 1/20 0.40
NOS2 P35228 1/20 0.40
AAK1 Q2M2I8 1/20 0.39
BACE1 P56817 1/20 0.39
KIF20B Q96Q89 1/20 0.39
ADRB2 P07550 1/20 0.39
NCF1 P14598 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPBWR1 P48145 1/20 0.38
KIF11 P52732 1/20 0.38
EGFR P00533 1/20 0.38
C1R P00736 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439770 0.87 BACE1 (0.42) CYP1A2CYP3A4CYP2C19NOS3NOS2
SCHEMBL437067 0.81 MAOB (0.46) PARP1MAOBNOS3NOS2BACE1
SCHEMBL438239 0.78 ACHE (0.46)
SCHEMBL442249 0.77 NPC1 (0.41) CYP1A2CYP3A4SMN1; SMN2KIF11NFKB1
SCHEMBL438818 0.76 ALDH1A1 (0.53) PARP1CYP1A2CYP2C19KDM4EALDH1A1
SCHEMBL29878151 0.75 ADRB2 (0.51) PARP1MAOBNOS3NOS2AAK1
SCHEMBL317413 0.75 ADRB2 (0.51) PARP1MAOBNOS3NOS2AAK1
SCHEMBL442268 0.75 ACHE (0.46) PARP1CYP3A4KDM4EALDH1A1SMN1; SMN2
SCHEMBL438932 0.75 ACHE (0.46) BACE1EGFR
SCHEMBL9591539 0.74 MAOB (0.46) PARP1MAOBAAK1KIF20BADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed