SCHEMBL440009

SCHEMBL440009

Cc1c(Cl)ccc2c(N)c(Br)cnc12

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.38
PDPK1 O15530 1/20 0.38
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
PKM P14618 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 2/20 0.33
THRB P10828 1/20 0.33
TP53 P04637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ALDH1A1 P00352 1/20 0.32
PPARA Q07869 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436942 0.84 HAVCR2 (0.41) HAVCR2PDPK1CCR1CCR5CCR8
SCHEMBL439739 0.84 CCR1 (0.39) HAVCR2CCR1CCR5CCR8MEN1
SCHEMBL437599 0.83 CCR1 (0.42) HAVCR2CCR1CCR5CCR8MEN1
SCHEMBL439423 0.83 HAVCR2 (0.36) HAVCR2MEN1KMT2AMAPTALDH1A1
SCHEMBL441974 0.80 HAVCR2 (0.38) HAVCR2PDPK1CCR1CCR5CCR8
SCHEMBL437260 0.76 HAVCR2 (0.67) HAVCR2PKMMEN1KMT2AMAPT
SCHEMBL441951 0.76 HAVCR2 (0.58) HAVCR2MEN1KMT2AMAPTALDH1A1
SCHEMBL436747 0.73 CYP3A4 (0.32) MEN1KMT2AMAPT
SCHEMBL436601 0.73 KMT2A (0.33) HAVCR2MEN1KMT2AALDH1A1
SCHEMBL441701 0.72 ALDH1A1 (0.43) HAVCR2PDPK1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed