SCHEMBL4407658

SCHEMBL4407658

COc1ccc(C(C)(C)C)cc1C(=O)Nc1ccc(C)c(-c2cc(C(=O)NCCc3cccnc3)on2)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CYP3A4 P08684 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
PTAFR P25105 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CYP1A2 P05177 2/20 0.41
MAPK1 P28482 1/20 0.41
TSHR P16473 1/20 0.41
BLM P54132 1/20 0.41
GAA P10253 1/20 0.40
CYP2C19 P33261 2/20 0.40
NAMPT P43490 1/20 0.40
ADRB3 P13945 1/20 0.40
BRAF P15056 1/20 0.39
LRRK2 Q5S007 2/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4419761 0.93 CYP1A2 (0.49) NPC1RAB9ACYP3A4MEN1KMT2A
SCHEMBL4412543 0.91 ALDH1A1 (0.42) NPC1RAB9ACYP3A4MEN1KMT2A
SCHEMBL4411700 0.85 MEN1 (0.43) CYP3A4MEN1KMT2ACYP1A2TSHR
SCHEMBL4551944 0.82 NR1H4 (0.46) MEN1KMT2ATSHRGAABRAF
SCHEMBL4417707 0.82 CYP3A4 (0.43) RAB9ACYP3A4MEN1KMT2AL3MBTL1
SCHEMBL4420074 0.81 RAF1 (0.49) NPC1RAB9AL3MBTL1BRAF
SCHEMBL14473103 0.81 MEN1 (0.46) NPC1RAB9ACYP3A4MEN1KMT2A
SCHEMBL4415213 0.79 RAF1 (0.45) NPC1RAB9AMEN1KMT2ABRAF
SCHEMBL4409369 0.79 RAB9A (0.51) NPC1RAB9AMEN1KMT2AL3MBTL1
SCHEMBL4410129 0.79 MEN1 (0.44) NPC1RAB9ACYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035005-A2 THERAPY USING CYTOKINE INHIBITORS Kemia, INC. (US) 2009-03-18 EP disclosed
WO-2007146712-A2 THERAPY USING CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-12-21 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed