SCHEMBL4417038

SCHEMBL4417038

CCCCNC(=O)Oc1cc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)n(CC2CCCCC2)c1C

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.39
HTR2A P28223 3/20 0.36
HTR2C P28335 3/20 0.36
SLC6A4 P31645 3/20 0.36
NCEH1 Q6PIU2 1/20 0.35
CNR2 P34972 1/20 0.35
CHRM4 P08173 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ACHE P22303 1/20 0.35
TRPV4 Q9HBA0 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4425227 0.92 CNR1 (0.41) CNR1HTR2AHTR2CSLC6A4NCEH1
SCHEMBL4417093 0.85 MAPT (0.43) CNR1HTR2AHTR2CSLC6A4NCEH1
SCHEMBL4423695 0.85 HTR2A (0.41) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL3919171 0.84 HTR2A (0.50) CNR1HTR2AHTR2CSLC6A4CHRM4
SCHEMBL4423191 0.84 NCEH1 (0.41) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL4425373 0.84 CNR1 (0.40) CNR1HTR2AHTR2CSLC6A4CNR2
SCHEMBL4418725 0.84 HTR2A (0.46) HTR2AHTR2CSLC6A4CNR2
SCHEMBL4419939 0.83 HTR2A (0.42) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL4423636 0.83 ALDH1A1 (0.47) CNR1HTR2AHTR2CSLC6A4CNR2
SCHEMBL4417423 0.82 MGLL (0.43) HTR2AHTR2CSLC6A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-B1 CB 1 RECEPTOUR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2009-12-02 EP claimed