SCHEMBL4417093

SCHEMBL4417093

CCCCNC(=O)Oc1cc(-c2ccc(F)cc2)n(CC2CCCCC2)c1C

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.43
NCEH1 Q6PIU2 1/20 0.42
HTR2A P28223 3/20 0.41
HTR2C P28335 3/20 0.41
SLC6A4 P31645 3/20 0.41
FAAH O00519 2/20 0.39
TSHR P16473 1/20 0.39
ACHE P22303 2/20 0.39
CNR1 P21554 2/20 0.38
CNR2 P34972 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MGLL Q99685 1/20 0.37
ABHD12 Q8N2K0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4423695 0.93 HTR2A (0.41) MAPTNCEH1HTR2AHTR2CSLC6A4
SCHEMBL4423191 0.91 NCEH1 (0.41) NCEH1HTR2AHTR2CSLC6A4TSHR
SCHEMBL4418725 0.91 HTR2A (0.46) HTR2AHTR2CSLC6A4FAAHCNR2
SCHEMBL4425227 0.90 CNR1 (0.41) NCEH1HTR2AHTR2CSLC6A4FAAH
SCHEMBL4419939 0.90 HTR2A (0.42) NCEH1HTR2AHTR2CSLC6A4FAAH
SCHEMBL4423636 0.90 ALDH1A1 (0.47) MAPTHTR2AHTR2CSLC6A4ACHE
SCHEMBL4419276 0.89 ACHE (0.39) MAPTNCEH1HTR2AHTR2CSLC6A4
SCHEMBL4417700 0.88 NCEH1 (0.42) NCEH1HTR2AHTR2CSLC6A4FAAH
SCHEMBL4422250 0.88 HTR2A (0.46) MAPTHTR2AHTR2CSLC6A4ACHE
SCHEMBL4417423 0.87 MGLL (0.43) MAPTHTR2AHTR2CSLC6A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-B1 CB 1 RECEPTOUR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2009-12-02 EP claimed