SCHEMBL4419939

SCHEMBL4419939

CCCCNC(=O)Oc1cc(-c2cccc(F)c2)n(CC2CCCCC2)c1C

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.42
HTR2C P28335 3/20 0.42
SLC6A4 P31645 3/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NCEH1 Q6PIU2 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ACHE P22303 1/20 0.38
FAAH O00519 2/20 0.37
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417093 0.90 MAPT (0.43) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL4429632 0.89 ALDH1A1 (0.43) HTR2AHTR2CSLC6A4ALDH1A1HSD17B10
SCHEMBL4423191 0.89 NCEH1 (0.41) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL4423695 0.86 HTR2A (0.41) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL4417700 0.86 NCEH1 (0.42) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL4417423 0.85 MGLL (0.43) HTR2AHTR2CSLC6A4ALDH1A1
SCHEMBL3918250 0.85 HTR2A (0.57) HTR2AHTR2CSLC6A4NPC1RAB9A
SCHEMBL4418725 0.85 HTR2A (0.46) HTR2AHTR2CSLC6A4FAAH
SCHEMBL4425227 0.84 CNR1 (0.41) HTR2AHTR2CSLC6A4NCEH1ALDH1A1
SCHEMBL4423636 0.84 ALDH1A1 (0.47) HTR2AHTR2CSLC6A4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-B1 CB 1 RECEPTOUR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2009-12-02 EP claimed