SCHEMBL4425227

SCHEMBL4425227

CCCCNC(=O)Oc1cc(-c2ccc(C(F)(F)F)cc2)n(CC2CCCCC2)c1C

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.41
MGLL Q99685 1/20 0.39
HTR2A P28223 4/20 0.39
HTR2C P28335 4/20 0.39
SLC6A4 P31645 4/20 0.39
ADAMTS4 O75173 1/20 0.38
ADAMTS5 Q9UNA0 1/20 0.38
TRPV4 Q9HBA0 1/20 0.37
NCEH1 Q6PIU2 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36
FAAH O00519 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417038 0.92 CNR1 (0.39) CNR1HTR2AHTR2CSLC6A4TRPV4
SCHEMBL4417093 0.90 MAPT (0.43) CNR1MGLLHTR2AHTR2CSLC6A4
SCHEMBL4423695 0.90 HTR2A (0.41) MGLLHTR2AHTR2CSLC6A4NCEH1
SCHEMBL4418725 0.88 HTR2A (0.46) HTR2AHTR2CSLC6A4FAAH
SCHEMBL4423636 0.88 ALDH1A1 (0.47) CNR1MGLLHTR2AHTR2CSLC6A4
SCHEMBL4423191 0.87 NCEH1 (0.41) MGLLHTR2AHTR2CSLC6A4NCEH1
SCHEMBL4419276 0.86 ACHE (0.39) MGLLHTR2AHTR2CSLC6A4NCEH1
SCHEMBL4422250 0.86 HTR2A (0.46) MGLLHTR2AHTR2CSLC6A4ALDH1A1
SCHEMBL4417423 0.85 MGLL (0.43) MGLLHTR2AHTR2CSLC6A4ALDH1A1
SCHEMBL3919639 0.85 HTR2A (0.53) CNR1HTR2AHTR2CSLC6A4TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-B1 CB 1 RECEPTOUR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2009-12-02 EP claimed