SCHEMBL4423636

SCHEMBL4423636

CCCCNC(=O)Oc1cc(-c2ccc(OC)cc2)n(CC2CCCCC2)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
CRHBP P24387 1/20 0.47
HTT P42858 1/20 0.47
CRHR2 Q13324 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HPGD P15428 2/20 0.44
TDP1 Q9NUW8 1/20 0.42
PLA2G2A P14555 1/20 0.42
MGLL Q99685 3/20 0.41
ACHE P22303 1/20 0.41
HTR2A P28223 3/20 0.40
HTR2C P28335 3/20 0.40
SLC6A4 P31645 3/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4423695 0.92 HTR2A (0.41) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL4429632 0.90 ALDH1A1 (0.43) ALDH1A1PLA2G2AHTR2AHTR2CSLC6A4
SCHEMBL4417423 0.90 MGLL (0.43) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL4418725 0.90 HTR2A (0.46) HTR2AHTR2CSLC6A4CNR2
SCHEMBL4417093 0.90 MAPT (0.43) ALDH1A1MAPTMGLLACHEHTR2A
SCHEMBL4419276 0.90 ACHE (0.39) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL4426602 0.89 PLA2G2A (0.42) ALDH1A1TDP1PLA2G2AMGLLACHE
SCHEMBL4425227 0.88 CNR1 (0.41) ALDH1A1MGLLACHEHTR2AHTR2C
SCHEMBL4422250 0.88 HTR2A (0.46) ALDH1A1MAPTKMT2AMEN1HPGD
SCHEMBL5048696 0.87 CDC25A (0.43) ALDH1A1MAPTKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-B1 CB 1 RECEPTOUR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2009-12-02 EP claimed