SCHEMBL442249

SCHEMBL442249

Nc1c(Cl)cnc2cc(OC(F)(F)F)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CYP2C9 P11712 2/20 0.41
SCN5A Q14524 2/20 0.41
GMNN O75496 1/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
ALOX15 P16050 1/20 0.41
NFKB1 P19838 1/20 0.41
SLC6A2 P23975 1/20 0.41
SCN4A P35499 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL437175 0.88 NPC1 (0.44) NPC1RAB9ACYP2C9SCN5AGMNN
SCHEMBL439912 0.82 ALOX5AP (0.42) NPC1RAB9ACYP2C9SCN5AGMNN
SCHEMBL440277 0.80 ACHE (0.50)
SCHEMBL9796693 0.77 KDM4E (0.42) NPC1RAB9ACYP2C9SCN5AGMNN
SCHEMBL30509463 0.77 KDM4E (0.42) NPC1RAB9ACYP2C9SCN5AGMNN
SCHEMBL438632 0.77 PARP1 (0.45) CYP1A2CYP3A4NFKB1SMN1; SMN2KIF11
SCHEMBL438239 0.74 ACHE (0.46)
SCHEMBL21143460 0.73 TRPA1 (0.44) SCN5ASCN9ATRPA1
SCHEMBL442268 0.71 ACHE (0.46) LMNATP53CYP3A4GAAALOX15
SCHEMBL438932 0.71 ACHE (0.46) JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed