SCHEMBL442268

SCHEMBL442268

Cc1ccc2c(N)c(Cl)cnc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.46
BCHE P06276 4/20 0.45
GRIN1 Q05586 4/20 0.45
GRIN2A Q12879 4/20 0.45
CHEK1 O14757 1/20 0.41
PARP1 P09874 1/20 0.41
PIM1 P11309 1/20 0.41
RPS6KA3 P51812 1/20 0.41
LMNA P02545 2/20 0.40
PLG P00747 1/20 0.39
PLAU P00749 1/20 0.39
PLAT P00750 1/20 0.39
HTR1A P08908 2/20 0.39
ADRA1D P25100 2/20 0.39
ADRA1A P35348 2/20 0.39
ADRA1B P35368 2/20 0.39
TNF P01375 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL440082 0.86 LMNA (0.47) ACHEBCHEGRIN1GRIN2APARP1
SCHEMBL12210442 0.81 ACHE (0.49) ACHEBCHEGRIN1GRIN2ACHEK1
SCHEMBL438932 0.79 ACHE (0.46) ACHEBCHEGRIN1GRIN2ATNF
SCHEMBL438239 0.79 ACHE (0.46) ACHEBCHEGRIN1GRIN2A
SCHEMBL437293 0.79 ACHE (0.43) ACHEBCHEGRIN1GRIN2ACHEK1
SCHEMBL440277 0.78 ACHE (0.50) ACHEBCHEPLGPLAUHTR1A
SCHEMBL441831 0.78 ALDH1A1 (0.46) ACHEBCHEGRIN1GRIN2ATNF
SCHEMBL436602 0.75 ACHE (0.44) ACHEPIM1ALDH1A1CYP3A4
SCHEMBL438632 0.75 PARP1 (0.45) PARP1KDM4EALDH1A1CYP3A4SMN1; SMN2
SCHEMBL437696 0.73 KDM4E (0.50) ACHEBCHEGRIN1GRIN2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed