SCHEMBL4462898

SCHEMBL4462898

CCCc1cc(Cc2c(N)nc(N)nc2N2CCN(S(C)(=O)=O)CC2)on1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
PIK3CA P42336 12/20 0.34
PIK3CB P42338 9/20 0.34
PIK3CD O00329 8/20 0.34
PIK3CG P48736 8/20 0.34
MTOR P42345 8/20 0.34
PIK3R1 P27986 7/20 0.34
DHFR P00374 2/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NUDT1 P36639 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4469774 0.84 NUDT1 (0.49) KDM4EPIK3CADHFRALDH1A1MAPT
SCHEMBL4462891 0.84 IGF1R (0.43) KDM4EPIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL4457078 0.69 IGF1R (0.41) ABL1BCR
SCHEMBL4457348 0.69 HRH3 (0.35)
SCHEMBL4463994 0.68 IGF1R (0.31)
SCHEMBL4469769 0.67 NUDT1 (0.46) KDM4EPIK3CAMTORDHFRMAPT
SCHEMBL4457095 0.62 DRD2 (0.42) KDM4ENPC1RAB9AALDH1A1MAPT
SCHEMBL26608009 0.61 ABL1 (0.50) KDM4ENPC1RAB9APIK3CAPIK3CB
SCHEMBL459183 0.60 PPARA (0.43) NPC1RAB9AALDH1A1HPGDSMN1; SMN2
SCHEMBL603299 0.60 HRH4 (0.51) NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed