SCHEMBL4495477

SCHEMBL4495477

CCc1c(C(=O)O)c(C=O)n(C)c1-c1ccc(C(=O)OC)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
ERN1 O75460 3/20 0.40
MAPT P10636 4/20 0.38
RAB9A P51151 1/20 0.38
DHFR P00374 1/20 0.38
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
AR P10275 1/20 0.37
SETD7 Q8WTS6 1/20 0.36
TSHR P16473 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4495795 0.86 ERN1 (0.46) ALDH1A1ERN1DHFRGLAHPGD
SCHEMBL4491009 0.83 ALDH1A1 (0.43) ALDH1A1MAPTRAB9AHTTHPGD
SCHEMBL4488870 0.80 MEN1 (0.43) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4498679 0.80 CCNC (0.36) ALDH1A1MAPTRAB9AHTTHPGD
SCHEMBL4492957 0.73 GRIA2 (0.42) ALDH1A1ERN1MAPTRAB9AMEN1
SCHEMBL4488653 0.70 ERCC1 (0.38) ALDH1A1MAPTRAB9AMEN1KMT2A
SCHEMBL4492339 0.69 MAPT (0.34) ALDH1A1MAPTRAB9AMEN1KMT2A
SCHEMBL4480912 0.68
SCHEMBL4496740 0.68 GRM5 (0.39) MAPTRAB9AMEN1KMT2AKDM4E
SCHEMBL4500631 0.68 DHODH (0.37) ALDH1A1DHFRHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed