SCHEMBL4495795

SCHEMBL4495795

CCc1c(C(=O)O)c(C=O)n(C)c1-c1cccc(C(=O)OC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.46
ALDH1A1 P00352 2/20 0.41
DHFR P00374 2/20 0.40
TGFBR1 P36897 1/20 0.39
HPGD P15428 2/20 0.39
GLA P06280 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4495477 0.86 ALDH1A1 (0.42) ERN1ALDH1A1DHFRHPGDGLA
SCHEMBL4491009 0.82 ALDH1A1 (0.43) ALDH1A1HPGDL3MBTL1POLB
SCHEMBL4498679 0.73 CCNC (0.36) ALDH1A1HPGDL3MBTL1POLB
SCHEMBL4488870 0.72 MEN1 (0.43) ALDH1A1
SCHEMBL4495792 0.70 ERN1 (0.47) ERN1ALDH1A1DHFRHPGDL3MBTL1
SCHEMBL4496740 0.70 GRM5 (0.39) TGFBR1TP53POLB
SCHEMBL4504195 0.70 CCR1 (0.38) ALDH1A1CNR1
SCHEMBL4488653 0.69 ERCC1 (0.38) ALDH1A1HPGDTDP1L3MBTL1POLB
SCHEMBL4485732 0.69 KMT2A (0.47) POLB
SCHEMBL3032014 0.69 KMO (0.63) ERN1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed