SCHEMBL4485732

SCHEMBL4485732

CCc1c(C(=O)O)c(C=O)n(Cc2ccccc2)c1-c1cccc(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.47
POLB P06746 1/20 0.46
PLA2G2A P14555 6/20 0.45
SLC16A3 O15427 1/20 0.43
SLC16A1 P53985 1/20 0.43
MCTS1 Q9ULC4 1/20 0.43
CCR2 P41597 1/20 0.42
EDNRB P24530 2/20 0.42
EDNRA P25101 1/20 0.42
PPARG P37231 2/20 0.41
FEN1 P39748 1/20 0.41
YWHAH Q04917 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
DRD4 P21917 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2C P28335 1/20 0.41
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4490040 0.88 GFER (0.47) PLA2G2AEDNRBFEN1PLA2G1B
SCHEMBL4494579 0.87 ALDH1A1 (0.43) KMT2APOLB
SCHEMBL4559832 0.86 TP53 (0.46) KMT2AFEN1
SCHEMBL4490747 0.86 PGR (0.43) KMT2APLA2G2ASLC16A3MCTS1CCR2
SCHEMBL4484664 0.82 CFTR (0.45) SLC16A3SLC16A1MCTS1CCR2FEN1
SCHEMBL4492983 0.82 ERCC5 (0.47) KMT2AFEN1
SCHEMBL4477472 0.82 PGR (0.48) KMT2APLA2G2ACCR2FEN1
SCHEMBL4482567 0.80 PLA2G2A (0.43) KMT2APLA2G2APLA2G1B
SCHEMBL4485664 0.79 KDM4E (0.40) KMT2APOLB
SCHEMBL4492336 0.77 AR (0.47) KMT2APOLBFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed