SCHEMBL4497714

SCHEMBL4497714

CCc1c(C(=O)O)c(C=O)n(C)c1-c1cccc(OC)n1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.40
BTK Q06187 1/20 0.36
CNR1 P21554 1/20 0.34
NR4A2 P43354 1/20 0.33
DHODH Q02127 1/20 0.33
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4496740 0.85 GRM5 (0.39)
SCHEMBL4492957 0.75 GRIA2 (0.42)
SCHEMBL4491009 0.75 ALDH1A1 (0.43) DHODH
SCHEMBL4504195 0.73 CCR1 (0.38) CNR1
SCHEMBL4495795 0.72 ERN1 (0.46) CNR1
SCHEMBL4498679 0.72 CCNC (0.36)
SCHEMBL4495477 0.71 ALDH1A1 (0.42)
SCHEMBL4488653 0.70 ERCC1 (0.38)
SCHEMBL4491753 0.70 POLB (0.35) DHODH
SCHEMBL4490745 0.69 GRIA2 (0.40) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed