SCHEMBL4518769

SCHEMBL4518769

CC(C)=Cc1ccccc1F

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 9/20 0.54
TRPA1 O75762 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
HIF1A Q16665 1/20 0.53
NPC1 O15118 1/20 0.47
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRIN2B Q13224 2/20 0.44
GRIN2C Q14957 2/20 0.44
GRIN3A Q8TCU5 2/20 0.44
ERN1 O75460 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2340381 0.82 LMNA (0.38) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL24832683 0.80 ERN1 (0.44) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL28178629 0.79 ALDH1A1 (0.53) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL23240183 0.79 TRPA1 (0.60) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL5203307 0.79 ALDH1A1 (0.53) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL30138202 0.78 NFE2L2 (0.56) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL13615662 0.78 NFE2L2 (0.56) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL149582 0.77 CYP1A2 (0.58) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL3402801 0.77 CYP1A2 (0.58) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9
SCHEMBL26552230 0.77 TRPA1 (0.46) NFE2L2TRPA1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220002663-A1 SELECTIVE SALMONELLA OR E. COLI CULTIVATION METHOD, COMPOSITIONS AND USES Solus Scientific Solutions Ltd (GB) 2022-01-06 US disclosed
EP-3115357-B1 BENZYLIDENEGUANIDINE DERIVATIVES AND THERAPEUTIC USE FOR THE TREATMENT OF PROTEIN MISFOLDING DISEASES RES & INNOVATION UK (GB) 2020-08-12 EP disclosed
EP-1736471-B1 3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES MITSUI CHEMICALS AGRO INC (JP) 2014-01-08 EP disclosed
US-7632783-B2 fungicides, pesticides for protecting rice crop, tomatoes, cucumbers and green beans; 3-(5-fluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quinoline MITSUI CHEMICALS AGRO, INC. (JP) 2009-12-15 US disclosed
US-20080275242-A1 3-(Dihydro(Tetrahydro)Isoquinolin-1-Yl)Quinoline Compound MITSUI CHEMICALS CROP & LIFE SOLUTIONS, INC. (JP) 2008-11-06 US disclosed
US-20080096894-A1 Anti-Bacterial Compounds ASTON UNIVERSITY (GB) 2008-04-24 US disclosed
US-20080096894-A1 Anti-Bacterial Compounds ASTON UNIVERSITY (GB) 2008-04-24 US disclosed
CN-1324015-C Pyridine and pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2007-07-04 CN disclosed
CN-1989101-A (Diaryl-methyl)-malononitriles and their use as estrogen receptor ligands WYETH CORP (US) 2007-06-27 CN disclosed
EP-1736471-A1 3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES Sankyo Agro Company, Limited (JP) 2006-12-27 EP disclosed
CN-1630644-A Novel pyridine and pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2005-06-22 CN disclosed
EP-0758328-B1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BTG INT LTD (GB) 2003-07-16 EP disclosed
EP-0667864-B1 TRICYCLIC COMPOUNDS WITH PHARMACEUTICAL ACTIVITY ZENECA LTD (GB) 1997-09-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080275242-A1 3-(Dihydro(Tetrahydro)Isoquinolin-1-Yl)Quinoline Compound QTRT1, RABL3, RECQL NFE2L2 1109/4885TRPA1 2092/4885CYP1A2 171/4885
US-20080096894-A1 Anti-Bacterial Compounds MRPL21, PGLS, FOSB NFE2L2 2689/4885TRPA1 2552/4885CYP1A2 3458/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.