SCHEMBL4531591

SCHEMBL4531591

O=C(NCCC1CCCN1S(=O)(=O)c1ccccc1Cl)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
P2RX7 Q99572 1/20 0.41
HSD11B1 P28845 3/20 0.41
HPGD P15428 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4542459 0.90 P2RX7 (0.42) P2RX7HSD11B1HPGD
SCHEMBL4531364 0.87 HSD11B1 (0.44) P2RX7HSD11B1HPGD
SCHEMBL4537550 0.84 PAX8 (0.56) DRD2DRD4
SCHEMBL4542139 0.83 PAX8 (0.45) DRD2DRD4
SCHEMBL4531594 0.82 TDP1 (0.42) DRD2HSD11B1TDP1HDAC3HDAC4
SCHEMBL4541325 0.82 HDAC3 (0.50) DRD2DRD4P2RX7HSD11B1HPGD
SCHEMBL4539750 0.81 HSD11B1 (0.52) HSD11B1
SCHEMBL4537477 0.80 NCOA1 (0.53) HPGD
SCHEMBL4537510 0.80 RAB9A (0.56) TDP1
SCHEMBL8066442 0.80 RAB9A (0.42) HSD11B1TDP1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed