SCHEMBL4537510

SCHEMBL4537510

O=C(NCCC1CCCN1S(=O)(=O)c1ccc(F)cc1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.56
NPC1 O15118 1/20 0.54
HTR7 P34969 2/20 0.49
MAPT P10636 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ATM Q13315 1/20 0.46
PAX8 Q06710 1/20 0.45
NCOA1 Q15788 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
LMNA P02545 1/20 0.44
TRPA1 O75762 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ENPP3 O14638 1/20 0.43
CA12 O43570 1/20 0.43
ENPP1 P22413 1/20 0.43
ENPP2 Q13822 1/20 0.43
CA9 Q16790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537550 0.90 PAX8 (0.56) RAB9AHTR7PAX8LMNAALDH1A1
SCHEMBL4537477 0.90 NCOA1 (0.53) RAB9ANPC1PAX8NCOA1NCOA3
SCHEMBL4535339 0.90 ATM (0.47) RAB9AHTR7ATMPAX8LMNA
SCHEMBL4536836 0.89 BRD4 (0.55) RAB9ANPC1PAX8NCOA1NCOA3
SCHEMBL4536842 0.87 RAB9A (0.50) RAB9ANPC1MAPTTDP1ATM
SCHEMBL4535463 0.83 HTR7 (0.55) RAB9ANPC1HTR7NCOA1NCOA3
SCHEMBL4542139 0.83 PAX8 (0.45) RAB9ANPC1HTR7PAX8SMN1; SMN2
SCHEMBL4537513 0.82 RAB9A (0.58) RAB9ANPC1HTR7MAPTTDP1
SCHEMBL4534658 0.81 CYP3A4 (0.49) MAPTSMN1; SMN2ALDH1A1ENPP3CA12
SCHEMBL4531591 0.80 DRD2 (0.42) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed