SCHEMBL4535199

SCHEMBL4535199

COc1ccc(S(=O)(=O)N2CCCCC2CC(=O)NC23CC4CC(CC(C4)C2)C3)cc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 8/20 0.53
MMP3 P08254 7/20 0.53
MMP7 P09237 6/20 0.53
MMP13 P45452 4/20 0.53
BDKRB1 P46663 1/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.49
PAX8 Q06710 1/20 0.49
MMP9 P14780 6/20 0.47
MMP2 P08253 5/20 0.47
MMP8 P22894 5/20 0.47
CNR2 P34972 1/20 0.47
HCRTR1 O43613 1/20 0.46
HCRTR2 O43614 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4542205 0.97 RAB9A (0.52) MMP1MMP3MMP7MMP13BDKRB1
SCHEMBL4540868 0.89 BDKRB1 (0.49) BDKRB1RAB9APAX8
SCHEMBL4537833 0.87 RAB9A (0.48) NPC1RAB9A
SCHEMBL4541294 0.87 PSEN1 (0.56) BDKRB1PAX8
SCHEMBL4537242 0.87 NPC1 (0.53) BDKRB1NPC1RAB9A
SCHEMBL4537185 0.87 RAB9A (0.56) MMP1MMP3MMP7MMP13NPC1
SCHEMBL4536688 0.86 FKBP1A (0.51) BDKRB1NPC1RAB9ACNR2HCRTR1
SCHEMBL4541024 0.86 RAB9A (0.48) BDKRB1RAB9APAX8
SCHEMBL4535169 0.86 HTR7 (0.54) BDKRB1RAB9ACNR2HCRTR1HCRTR2
SCHEMBL4539776 0.85 BRD4 (0.53) BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed