SCHEMBL4550682

SCHEMBL4550682

COc1ccc(-c2cccc3[nH]c(OC(=O)NC4CCN(CCN5C6CCC5CC(O)C6)CC4)cc23)cn1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.39
TLR9 Q9NR96 1/20 0.39
PIK3CA P42336 6/20 0.37
CD274 Q9NZQ7 1/20 0.36
ATM Q13315 2/20 0.36
DYRK1A Q13627 2/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
MTOR P42345 2/20 0.35
EGLN1 Q9GZT9 1/20 0.35
HTR7 P34969 1/20 0.34
WNT1 P04628 1/20 0.34
ACKR3 P25106 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4403763 0.92 TLR9 (0.42) GSK3BTLR9PIK3CACD274ATM
SCHEMBL4398653 0.90 MCHR1 (0.37) GSK3BDYRK1A
SCHEMBL4396957 0.89 TLR9 (0.42) GSK3BTLR9CD274DYRK1AEGLN1
SCHEMBL916126 0.88 GSK3B (0.42) GSK3BTLR9PIK3CACD274DYRK1A
SCHEMBL4410357 0.86 GSK3B (0.40) GSK3BTLR9PIK3CACD274DYRK1A
SCHEMBL4551165 0.81 SIGMAR1 (0.40) TLR9CD274DYRK1A
SCHEMBL4401911 0.80 HTR1A (0.38) HTR7
SCHEMBL914569 0.80 TLR9 (0.44) GSK3BTLR9CD274DYRK1AEGLN1
SCHEMBL4403446 0.79 DYRK1A (0.37) GSK3BTLR9CD274DYRK1AWNT1
SCHEMBL4411339 0.78 HTR7 (0.38) DYRK1AHTR7WNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed