SCHEMBL4398653

SCHEMBL4398653

COc1ccc(-c2cccc3[nH]c(OC(=O)NC4CCN(CCN5C6CCC5CC(O)C6)CC4)cc23)cc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.37
SIGMAR1 Q99720 4/20 0.37
PLD2 O14939 1/20 0.36
PLD1 Q13393 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
KMT2A Q03164 1/20 0.36
DRD4 P21917 1/20 0.36
DYRK1A Q13627 1/20 0.35
CCR5 P51681 1/20 0.35
GSK3B P49841 1/20 0.35
CHRM3 P20309 1/20 0.35
CHRM1 P11229 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SLC2A1 P11166 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4551165 0.91 SIGMAR1 (0.40) MCHR1SIGMAR1KMT2ADRD4DYRK1A
SCHEMBL4550682 0.90 GSK3B (0.39) DYRK1AGSK3B
SCHEMBL4396992 0.88 KMT2A (0.41) MCHR1SIGMAR1KMT2ADRD4DYRK1A
SCHEMBL914281 0.88 DRD4 (0.41) PLD2PLD1KMT2ADRD4DYRK1A
SCHEMBL6966091 0.88 DRD4 (0.41) PLD2PLD1KMT2ADRD4DYRK1A
SCHEMBL4411339 0.83 HTR7 (0.38) KMT2ADYRK1A
SCHEMBL4541737 0.82 SLC2A1 (0.39) MCHR1SIGMAR1KMT2ADRD4DYRK1A
SCHEMBL4401911 0.81 HTR1A (0.38)
SCHEMBL4403763 0.81 TLR9 (0.42) DYRK1AGSK3B
SCHEMBL4396457 0.80 HRH3 (0.42) HRH3KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed