SCHEMBL4569989

SCHEMBL4569989

CCN1CCCC1CNC(=O)c1cc(-c2cc(NC(=O)c3cc(C(C)(C)C)cc(C#N)c3OC)ccc2C)no1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43
DRD3 P35462 1/20 0.43
RAB9A P51151 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4420133 0.88 RAB9A (0.48) KDM4EALDH1A1CYP1A2RAB9A
SCHEMBL4414341 0.88 USP30 (0.40) RAB9A
SCHEMBL4416983 0.86 RAB9A (0.41) DRD2KDM4EALDH1A1RAB9AABCG2
SCHEMBL4411132 0.84 BRAF (0.38) CYP1A2CYP3A4
SCHEMBL4412696 0.83 USP30 (0.40)
SCHEMBL4565792 0.80 MAPT (0.41) ALDH1A1CYP1A2CYP3A4RAB9A
SCHEMBL4413451 0.80 RAF1 (0.36)
SCHEMBL4410129 0.80 MEN1 (0.44) KDM4EALDH1A1CYP1A2CYP3A4MAPK1
SCHEMBL4411278 0.80 MAPT (0.37) KDM4EALDH1A1CYP1A2CYP3A4RAB9A
SCHEMBL4730519 0.79 ABCG2 (0.45) DRD2KDM4EALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035005-A2 THERAPY USING CYTOKINE INHIBITORS Kemia, INC. (US) 2009-03-18 EP disclosed
WO-2007146712-A2 THERAPY USING CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-12-21 WO disclosed