Water

Water

SCHEMBL460840

O.O=C1CCC(=O)c2ccccc21.O=C1CCC(=O)c2ccccc21

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 3/20 0.47
THRB known ✓ P10828 1/20 0.45
GSK3B known ✓ P49841 1/20 0.41
TYMS known ✓ P04818 1/20 0.41
PARP1 known ✓ P09874 1/20 0.39
MAOA P21397 4/20 0.54
MAOB P27338 2/20 0.54
CYP2A6 P11509 1/20 0.54
CES1 P23141 3/20 0.48
KMT2A Q03164 3/20 0.47
CDC25B P30305 2/20 0.47
S100A4 P26447 2/20 0.45
BCHE P06276 2/20 0.45
KDM4E B2RXH2 1/20 0.45
CES2 O00748 1/20 0.45
APAF1 O14727 1/20 0.45
TERT O14746 1/20 0.45
NPC1 O15118 1/20 0.45
PLIN1 O60240 1/20 0.45
TDP2 O95551 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL855431 0.97 MAOA (0.56) MAOAMAOBCYP2A6CES1MEN1
SCHEMBL29385474 0.97 MAOA (0.56) MAOAMAOBCYP2A6CES1MEN1
SCHEMBL2686810 0.82 CES1 (0.62) MAOAMAOBCYP2A6CES1BCHE
SCHEMBL31157901 0.82 CES1 (0.62) MAOAMAOBCYP2A6CES1BCHE
Acetic Acid SCHEMBL29684240 0.82 NOTUM (0.52) MAOAMAOBCYP2A6CES1MEN1
SCHEMBL29353311 0.80 MAOA (0.74) MAOAMAOBCYP2A6CES1BCHE
SCHEMBL1268680 0.80 MAOA (0.74) MAOAMAOBCYP2A6CES1BCHE
SCHEMBL24746 0.80 MAOA (0.74) MAOAMAOBCYP2A6CES1BCHE
SCHEMBL31454252 0.78 MAOA (0.71) MAOAMAOBCYP2A6CES1BCHE
SCHEMBL16552853 0.78 MAOA (0.71) MAOAMAOBCYP2A6CES1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9045654-B2 Multilayer articles capable of forming color images 3M INNOVATIVE PROPERTIES COMPANY (US) 2015-06-02 US claimed
US-8411120-B2 Generation of color images 3M INNOVATIVE PROPERTIES COMPANY (US) 2013-04-02 US claimed
US-20110121557-A1 MULTILAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY 2011-05-26 US claimed
US-20110063392-A1 GENERATION OF COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY 2011-03-17 US claimed
EP-2280823-A2 GENERATION OF COLOR IMAGES 3M Innovative Properties Company (US) 2011-02-09 EP claimed
WO-2009140088-A1 MULTI-LAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY (US) 2009-11-19 WO claimed
WO-2009140083-A2 GENERATION OF COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY (US) 2009-11-19 WO claimed
EP-2588317-B1 MULTI-LAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES AND METHODS OF FORMING COLOR IMAGES 3M INNOVATIVE PROPERTIES CO (US) 2020-03-18 EP disclosed
US-9045654-B2 Multilayer articles capable of forming color images 3M INNOVATIVE PROPERTIES COMPANY (US) 2015-06-02 US disclosed
US-8975012-B2 Multi-layer articles capable of forming color images and methods of forming color images 3M INNOVATIVE PROPERTIES COMPANY (US) 2015-03-10 US disclosed
US-8975011-B2 Multi-layer articles capable of forming color images and method of forming color images 3M INNOVATIVE PROPERTIES COMPANY (US) 2015-03-10 US disclosed
EP-2588317-A2 MULTI-LAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES AND METHODS OF FORMING COLOR IMAGES 3M Innovative Properties Company (US) 2013-05-08 EP disclosed
EP-2588316-A2 MULTI-LAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES AND METHODS OF FORMING COLOR IMAGES 3M Innovative Properties Company (US) 2013-05-08 EP disclosed
WO-2012012118-A2 MULTI-LAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES AND METHODS OF FORMING COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-01-26 WO disclosed
WO-2012003247-A2 MULTI-LAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES AND METHODS OF FORMING COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-01-05 WO disclosed
US-20110121557-A1 MULTILAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY 2011-05-26 US disclosed
US-20110063392-A1 GENERATION OF COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY 2011-03-17 US disclosed
EP-2280823-A2 GENERATION OF COLOR IMAGES 3M Innovative Properties Company (US) 2011-02-09 EP disclosed
WO-2009140088-A1 MULTI-LAYER ARTICLES CAPABLE OF FORMING COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY (US) 2009-11-19 WO disclosed
WO-2009140083-A2 GENERATION OF COLOR IMAGES 3M INNOVATIVE PROPERTIES COMPANY (US) 2009-11-19 WO disclosed