Water

Water

SCHEMBL4609376

CC(C)(N)c1ccccc1.O

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 1/20 0.44
ESR1 known ✓ P03372 2/20 0.42
ESR2 known ✓ Q92731 2/20 0.42
KCNN4 O15554 4/20 0.55
TAAR1 Q96RJ0 2/20 0.50
AKT1 P31749 1/20 0.50
AKT2 P31751 1/20 0.50
MAPK1 P28482 1/20 0.48
ALDH1A1 P00352 3/20 0.48
TSHR P16473 2/20 0.48
PDE2A O00408 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
ALOX15 P16050 1/20 0.44
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5872061 0.97 KCNN4 (0.52) KCNN4TAAR1AKT1AKT2MAPK1
Hydrochloric Acid SCHEMBL8388827 0.97 KCNN4 (0.52) KCNN4TAAR1AKT1AKT2MAPK1
Hydrochloric Acid SCHEMBL8387706 0.97 KCNN4 (0.52) KCNN4TAAR1AKT1AKT2MAPK1
SCHEMBL6145 0.97 KCNN4 (0.58) KCNN4TAAR1AKT1AKT2MAPK1
Bromide SCHEMBL414533 0.94 KCNN4 (0.55) KCNN4TAAR1AKT1AKT2MAPK1
Methylamine SCHEMBL20916863 0.94 KCNN4 (0.55) KCNN4TAAR1AKT1AKT2MAPK1
Fluoride SCHEMBL634655 0.94 KCNN4 (0.55) KCNN4TAAR1AKT1AKT2MAPK1
Iodide SCHEMBL6672017 0.94 KCNN4 (0.55) KCNN4TAAR1AKT1AKT2MAPK1
Hydrochloric Acid SCHEMBL8387827 0.94 KCNN4 (0.55) KCNN4TAAR1AKT1AKT2MAPK1
Bromide SCHEMBL3629993 0.94 KCNN4 (0.55) KCNN4TAAR1AKT1AKT2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 111 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12419942-B2 Use of the Salmonella spp type III secretion proteins as a protective vaccination UNIVERSITY OF KANSAS (US) 2025-09-23 US disclosed
CN-119730834-A Personal care compositions containing spherical silicone elastomer fine particles 迈图高新材料公司 2025-03-28 CN disclosed
US-12201715-B2 Personal care composition containing spherical silicone elastomer fine particles MOMENTIVE PERFORMANCE MATERIALS INC. (US) 2025-01-21 US disclosed
US-12102679-B2 FcRn-targeted therapeutics for the treatment of antibody-mediated autoimmune and albumin-mediated disease UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2024-10-01 US disclosed
WO-2024039563-A1 PERSONAL CARE COMPOSITION CONTAINING SPHERICAL SILICONE ELASTOMER FINE PARTICLES MOMENTIVE PERFORMANCE MATERIALS INC. (US) 2024-02-22 WO disclosed
US-20240058255-A1 PERSONAL CARE COMPOSITION CONTAINING SPHERICAL SILICONE ELASTOMER FINE PARTICLES MOMENTIVE PERFORMANCE MATERIALS INC. 2024-02-22 US disclosed
US-20230181723-A1 FcRn-TARGETED THERAPEUTICS FOR THE TREATMENT OF ANTIBODY-MEDIATED AUTOIMMUNE AND ALBUMIN-MEDIATED DISEASE UNIVERSITY OF MARYLAND, COLLEGE PARK 2023-06-15 US disclosed
CN-114470198-B IgY spray of SARS-CoV-2 egg yolk neutralization antibody for preventing and treating new coronal pneumonia 上海博满生物科技有限公司 2023-05-05 CN disclosed
US-20230136602-A1 Use of the Salmonella SPP Type III Secretion Proteins as a Protective Vaccination UNIVERSITY OF KANSAS 2023-05-04 US disclosed
CN-115667339-A Aqueous polyurethane resin dispersion 爱克发有限公司 2023-01-31 CN disclosed
WO-1998038859-A1 SULFONYL DIVALENT ARYL OR HETEROARYL HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998039316-A1 N-HYDROXY 4-SULFONYL BUTANAMIDE COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998039315-A1 AROMATIC SULFONYL ALPHA-CYCLOAMINO HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998039313-A1 THIOARYL SULFONAMIDE HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998039326-A1 AROMATIC SULFONYL ALPHA-HYDROXY HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed
EP-0482480-B1 Surface-treating agent and surface-treated EPDM article TOSHIBA SILICONE (JP) 1995-01-11 EP disclosed
EP-0482480-A1 Surface-treating agent and surface-treated EPDM article TOSHIBA SILICONE CO., LTD. (JP) 1992-04-29 EP disclosed
EP-0469613-A2 Organopolysiloxane/acrylate ester copolymer emulsion Dow Corning Toray Silicone Company, Limited (JP) 1992-02-05 EP disclosed
US-4622335-A AGRICULTURE BAYER AKTIENGESELLSCHAFT (DE) 1986-11-11 US disclosed