SCHEMBL4669567

SCHEMBL4669567

O=C(OCc1ccccc1)C1CCN1C(c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 10/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
CYP2C19 P33261 1/20 0.45
PREP P48147 1/20 0.44
AGTR2 P50052 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7064400 0.88 FKBP1A (0.50) FKBP1ASMN1; SMN2NPC1RAB9APREP
SCHEMBL7064334 0.86 FKBP1A (0.48) FKBP1ASMN1; SMN2NPC1RAB9APREP
SCHEMBL5785042 0.84 CACNA1A (0.57) SMN1; SMN2NPC1RAB9A
SCHEMBL10579873 0.84 FKBP1A (0.54) FKBP1ASMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL7066507 0.81 FKBP1A (0.47) FKBP1ASMN1; SMN2NPC1RAB9APREP
SCHEMBL2770710 0.81 KMT2A (0.48) CYP2C19AGTR2
SCHEMBL7062463 0.80 CCR1 (0.46) FKBP1A
SCHEMBL7066355 0.80 FKBP1A (0.47) FKBP1APREP
SCHEMBL5685743 0.79 ALDH1A1 (0.47) AGTR2
SCHEMBL5685826 0.79 ALDH1A1 (0.47) AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-56032454-A None JP disclosed
EP-1193253-B1 PROCESS FOR PRODUCING OPTICALLY ACTIVE AZETIDINE-2-CARBOXYLIC ACIDS KANEKA CORP (JP) 2008-06-25 EP disclosed
EP-1927588-A2 Process for producing optically active azetidine-2-carboxylic acids KANEKA CORPORATION (JP) 2008-06-04 EP disclosed
US-7262308-B2 Process for producing optically active azetidine-2-carboxylic acids KANEKA CORPORATION (JP) 2007-08-28 US disclosed
US-20050043547-A1 Process for producing optically active azetidine-2-carboxylic acids HONDA TATSUYA (JP) 2005-02-24 US disclosed
US-6838567-B1 Process for producing optically active azetidine-2-carboxylic acids KANEKA CORPORATION (JP) 2005-01-04 US disclosed
US-20040171849-A1 Process for producing optically active azetidine-2-carboxylic acid KANEKA CORPORATION (JP) 2004-09-02 US disclosed
EP-1415985-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE AZETIDINE-2-CARBOXYLIC ACID KANEKA CORPORATION (JP) 2004-05-06 EP disclosed
EP-0992491-B1 PROCESSES FOR PRODUCING AZETIDINE-2-CARBOXYLIC ACID AND INTERMEDIATES THEREOF KANEKA CORP (JP) 2003-03-05 EP disclosed
EP-0950057-B1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LAB (US) 2002-11-13 EP disclosed
US-6150535-A Processes for producing azetidine-2-carboxylic acid and intermediates thereof KANEKA CORPORATION (JP) 2000-11-21 US disclosed
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
US-6133253-A NEURONAL CELL DEATH PREVENTORS AND ANTI-INFLAMMATORIES ABBOTT LABORATORIES (US) 2000-10-17 US disclosed
EP-0992491-A1 PROCESSES FOR PRODUCING AZETIDINE-2-CARBOXYLIC ACID AND INTERMEDIATES THEREOF KANEKA CORPORATION (JP) 2000-04-12 EP disclosed
EP-0950057-A1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS Abbott Laboratories (US) 1999-10-20 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed
WO-1998025920-A1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LABORATORIES (US) 1998-06-18 WO disclosed
US-4349547-A Suppressing obesity and over-secretion of insulin with 2-(α-hydroxy-m-trifluoromethylbenzyl)azetidine TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1982-09-14 US disclosed
EP-0025880-A1 Azetidine derivative, its production, the derivative for use as an anti-obesity agent Takeda Chemical Industries, Ltd. (JP) 1981-04-01 EP disclosed
JP-S5632454-A AZETIDINE DERIVATIVE TAKEDA CHEM IND LTD 1981-04-01 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040171849-A1 Process for producing optically active azetidine-2-carboxylic acid HBB, ADCY2, ADCY9 FKBP1A 2054/4885SMN1; SMN2 1956/4885NPC1 2874/4885
US-20050043547-A1 Process for producing optically active azetidine-2-carboxylic acids AZI2, ALAD, HBB FKBP1A 1857/4885SMN1; SMN2 2424/4885NPC1 4418/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.