SCHEMBL4672123

SCHEMBL4672123

COc1ccc(CCCn2nnn(-c3ccc(C(N)=O)cc3)c2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 3/20 0.46
PARP10 Q53GL7 2/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
PARP1 P09874 1/20 0.46
PARP2 Q9UGN5 1/20 0.46
PARP4 Q9UKK3 1/20 0.46
DRD2 P14416 1/20 0.45
ALDH1A1 P00352 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
TP53 P04637 2/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
GFER P55789 1/20 0.43
VNN1 O95497 1/20 0.41
PTGDR Q13258 1/20 0.40
NPBWR1 P48145 1/20 0.39
MAP4K4 O95819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4672126 0.86 NPBWR1 (0.42) DRD2SMN1; SMN2LMNAMAPTNPBWR1
SCHEMBL4673352 0.85 MAPK1 (0.50) PARP1PARP2ALDH1A1HPGDTSHR
SCHEMBL4672086 0.80 KCNJ1 (0.53) ALDH1A1SMN1; SMN2LMNAMAPTHPGD
SCHEMBL4675102 0.77 ALDH1A1 (0.42) PARP10ALDH1A1SMN1; SMN2HPGDTSHR
SCHEMBL4670479 0.77 ALDH1A1 (0.39) MAPKAPK2PARP10ALDH1A1SMN1; SMN2HPGD
SCHEMBL6300283 0.77 PARP10 (0.47) PARP10TSHR
SCHEMBL4670081 0.73 ADRB2 (0.42) PARP10PARP2ALDH1A1TSHR
Water SCHEMBL4673066 0.72 ADRB2 (0.41) PARP10PARP2ALDH1A1TSHR
SCHEMBL4670046 0.72 PARP10 (0.40) PARP10PARP2ALDH1A1TSHRKDM4E
SCHEMBL4670624 0.72 PARP15 (0.40) PARP10PARP2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054881-B1 NOVEL SULFONAMIDE SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER CORP (US) 2008-07-30 EP disclosed